SCHEMBL11344285

SCHEMBL11344285

Cc1ccc2c(c1)CC(=O)c1cc(C(C)C(=O)OCCOCCO)ccc1O2

nearest known ligand 0.40

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 2/20 0.33
ABCC4 O15439 1/20 0.33
PTGS2 P35354 1/20 0.31
OPRK1 P41145 1/20 0.31
PDE4D Q08499 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11333573 0.90 PTGS2 (0.36) PTGS1ABCC4PTGS2OPRK1PDE4D
SCHEMBL29481375 0.84 LMNA (0.38)
SCHEMBL11339277 0.83 PTGS2 (0.48) PTGS1PTGS2OPRK1PDE4D
SCHEMBL11332871 0.82 YWHAG (0.36)
Bermoprofen SCHEMBL29454489 0.80 PTGS1 (0.49) PTGS1ABCC4PTGS2OPRK1PDE4D
Bermoprofen SCHEMBL25434 0.80 PTGS1 (0.49) PTGS1ABCC4PTGS2OPRK1PDE4D
SCHEMBL14434968 0.80 PTGS1 (0.41) PTGS1ABCC4PTGS2OPRK1PDE4D
SCHEMBL13875314 0.79 PTGS1 (0.38) PTGS1ABCC4PTGS2OPRK1PDE4D
Bermoprofen SCHEMBL11441448 0.78 PTGS1 (0.39) PTGS1ABCC4PTGS2OPRK1PDE4D
SCHEMBL11473894 0.77 PTGS2 (0.40) PTGS1ABCC4PTGS2OPRK1PDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0003893-B1 NOVEL DIBENZ (B,F) OXEPIN AND DIBENZO (B,F) THIEPIN COMPOUNDS AND PHARMACEUTICALLY ACCEPTABLE SALTS THEREOF, PROCESSES FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM Dainippon Pharmaceutical Co., Ltd. (JP) 1981-11-04 EP claimed
US-4238620-A ANTIPYRETICS; ANALGESICS; ANTIINFLAMMATORY AGENTS DAINIPPON PHARMACEUTICAL CO., LTD. (JP) 1980-12-09 US claimed
US-4238620-A ANTIPYRETICS; ANALGESICS; ANTIINFLAMMATORY AGENTS DAINIPPON PHARMACEUTICAL CO., LTD. (JP) 1980-12-09 US disclosed
EP-0003893-A1 Novel dibenz (b,f) oxepin and dibenzo (b,f) thiepin compounds and pharmaceutically acceptable salts thereof, processes for their preparation and pharmaceutical compositions containing them Dainippon Pharmaceutical Co., Ltd. (JP) 1979-09-05 EP disclosed