SCHEMBL1136899

SCHEMBL1136899

CC(C)(C)N(Cc1ccc(-c2cnccc2Oc2ccc([N+](=O)[O-])cc2F)cc1)C(=O)O

nearest known ligand 0.40

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.39
MAPT P10636 1/20 0.39
MAPK1 P28482 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
MET P08581 3/20 0.37
CYP19A1 P11511 6/20 0.37
CYP11B1 P15538 6/20 0.37
CYP11B2 P19099 6/20 0.37
HSPB1 P04792 2/20 0.37
S1PR4 O95977 1/20 0.37
TTR P02766 1/20 0.35
POLB P06746 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1136902 1.00 ALDH1A1 (0.39) ALDH1A1MAPTMAPK1L3MBTL1MET
SCHEMBL1137010 0.84 HSPB1 (0.41) ALDH1A1MAPTMAPK1L3MBTL1MET
SCHEMBL2257136 0.82 MMP13 (0.41) ALDH1A1MAPTMAPK1L3MBTL1MET
SCHEMBL2257142 0.82 MMP13 (0.41) ALDH1A1MAPTMAPK1L3MBTL1MET
SCHEMBL1137142 0.82 SLC22A12 (0.41) ALDH1A1MAPTMAPK1L3MBTL1MET
SCHEMBL28770683 0.81 MET (0.36) ALDH1A1MAPTMAPK1L3MBTL1MET
SCHEMBL12363119 0.81 NAMPT (0.41) ALDH1A1MAPTMAPK1L3MBTL1MET
SCHEMBL14045145 0.80 HSPB1 (0.50) ALDH1A1MAPTMAPK1L3MBTL1MET
SCHEMBL1137649 0.79 CYP11B1 (0.41) ALDH1A1MAPTMETCYP19A1CYP11B1
SCHEMBL1137363 0.79 POLB (0.42) ALDH1A1MAPTMAPK1L3MBTL1MET

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1737451-B1 MONOCYCLIC HETEROCYCLES AS KINASE INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2011-02-23 EP disclosed