SCHEMBL11380495

SCHEMBL11380495

O=C1CCc2c(OCC3CO3)ccc(OCCO)c2N1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.36
GLA P06280 1/20 0.36
PDE1A P54750 1/20 0.33
PDE1B Q01064 1/20 0.33
PDE4D Q08499 1/20 0.33
PDE7A Q13946 1/20 0.33
PDE1C Q14123 1/20 0.33
PDE7B Q9NP56 1/20 0.33
ADRB3 P13945 1/20 0.33
HTR2A P28223 2/20 0.33
SLC6A4 P31645 2/20 0.33
KDM4E B2RXH2 1/20 0.33
KMT2A Q03164 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
LMNA P02545 1/20 0.32
GAA P10253 1/20 0.32
PKM P14618 1/20 0.32
TP53 P04637 1/20 0.32
CYP3A4 P08684 1/20 0.32
TSHR P16473 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11381634 0.88 ALDH1A1 (0.39) ALDH1A1GLAADRB3HTR2ASLC6A4
SCHEMBL9385939 0.84 ALDH1A1 (0.41) ALDH1A1GLAADRB3HTR2ASLC6A4
SCHEMBL9534845 0.84 VDR (0.41) ALDH1A1GLAADRB3HTR2ASLC6A4
SCHEMBL9384498 0.83 ALDH1A1 (0.46) ALDH1A1GLAADRB3HTR2ASLC6A4
SCHEMBL9654091 0.83 ALDH1A1 (0.39) ALDH1A1GLAHTR2ASLC6A4TDP1
SCHEMBL11378856 0.82 ALDH1A1 (0.35) ALDH1A1GLAADRB3HTR2ASLC6A4
SCHEMBL9652974 0.81 ALDH1A1 (0.38) ALDH1A1GLAADRB3HTR2ASLC6A4
SCHEMBL9651024 0.81 HTR2A (0.44) ALDH1A1GLAADRB3HTR2ASLC6A4
SCHEMBL7091814 0.81 BRD4 (0.42) ALDH1A1GLAPDE4DTDP1
SCHEMBL6074729 0.81 BRD4 (0.42) ALDH1A1GLAPDE4DTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4289883-A ADRENERGIC BLOCKING AGENTS OF EXCELLENT CARDIOSELECTIVITY OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1981-09-15 US disclosed