SCHEMBL11394433

SCHEMBL11394433

COc1ccc(CC(=O)N(C)C2CCCCC2)cc1

nearest known ligand 0.64

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 3/20 0.64
CCR5 P51681 4/20 0.61
EPHX2 P34913 1/20 0.58
PTGDR2 Q9Y5Y4 1/20 0.50
TRPM8 Q7Z2W7 2/20 0.49
MEN1 O00255 2/20 0.49
KMT2A Q03164 2/20 0.49
NPC1 O15118 2/20 0.49
RAB9A P51151 2/20 0.49
SMN1; SMN2 Q16637 2/20 0.49
ALDH1A1 P00352 1/20 0.47
POLB P06746 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2405257 0.93 CCR5 (0.62) SIGMAR1CCR5EPHX2PTGDR2SMN1; SMN2
SCHEMBL5860907 0.86 CCR5 (0.56) SIGMAR1CCR5EPHX2PTGDR2SMN1; SMN2
SCHEMBL31473504 0.86 CCR5 (0.56) SIGMAR1CCR5EPHX2PTGDR2SMN1; SMN2
SCHEMBL14297341 0.84 NPC1 (0.55) SIGMAR1CCR5MEN1KMT2ANPC1
SCHEMBL3528763 0.83 SIGMAR1 (0.72) SIGMAR1CCR5EPHX2MEN1KMT2A
SCHEMBL2575803 0.82 MEN1 (0.51) SIGMAR1CCR5MEN1KMT2A
Hydrochloric Acid SCHEMBL11534945 0.82 SIGMAR1 (0.70) SIGMAR1CCR5EPHX2SMN1; SMN2ALDH1A1
SCHEMBL4283829 0.82 CCR5 (0.62) SIGMAR1CCR5EPHX2KMT2AALDH1A1
SCHEMBL5862792 0.79 KCNH2 (0.72) SIGMAR1CCR5
SCHEMBL15962426 0.78 SIGMAR1 (1.00) SIGMAR1MEN1KMT2ARAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4248877-A ANTIDEPRESSANTS, ANALGESICS, ANTIMIGRAINE AGENTS SANDOZ LTD. (CH) 1981-02-03 US disclosed
US-4178377-A USE TO TREAT PAIN AND MIGRAINE SANDOZ LTD. (CH) 1979-12-11 US disclosed