SCHEMBL11399009

SCHEMBL11399009

O=C1C[N+]([O-])=C(c2ccccc2F)c2cc(Br)ccc2N1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 3/20 0.57
GABRA5 P31644 3/20 0.57
GABRA3 P34903 3/20 0.57
GABRA2 P47869 3/20 0.57
GABRB2 P47870 2/20 0.57
GABRG2 P18507 1/20 0.42
GABRB3 P28472 1/20 0.42
CCNB2 O95067 4/20 0.41
CDK1 P06493 4/20 0.41
CCNB1 P14635 4/20 0.41
GSK3B P49841 4/20 0.41
CDK5 Q00535 4/20 0.41
CDK5R1 Q15078 4/20 0.41
CCNB3 Q8WWL7 4/20 0.41
KMT2A Q03164 5/20 0.40
MEN1 O00255 4/20 0.40
LMNA P02545 2/20 0.40
ADRA1A P35348 1/20 0.40
TGM2 P21980 1/20 0.38
CES1 P23141 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11319239 0.85 LMNA (0.57) GABRA1GABRA5GABRA3GABRA2GABRB2
SCHEMBL2846056 0.84 KMT2A (0.47) GABRA1GABRA5GABRA3GABRA2GABRB2
SCHEMBL10675729 0.82 SMN1; SMN2 (0.39) GABRA1GABRA5GABRA3GABRA2GABRB2
SCHEMBL7551382 0.72 NSD2 (0.40) KMT2AMEN1LMNATGM2CES1
SCHEMBL7548596 0.72 DAO (0.40) LMNAMAPTSMN1; SMN2NPC1ALDH1A1
SCHEMBL32681120 0.72 GABRA1 (0.55) GABRA1GABRA5GABRA3GABRA2GABRB2
SCHEMBL638723 0.72 GABRA1 (1.00) GABRA1GABRA5GABRA3GABRA2GABRB2
SCHEMBL6527541 0.72 GABRA1 (0.55) GABRA1GABRA5GABRA3GABRA2GABRB2
SCHEMBL31696096 0.72 GABRA1 (1.00) GABRA1GABRA5GABRA3GABRA2GABRB2
SCHEMBL7548112 0.70 MEN1 (0.33) KMT2AMEN1MAPTALDH1A1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4246270-A TRANQUILIZERS, MUSCLE RELAXANTS, AND SEDATIVES E. I. DU PONT DE NEMOURS AND COMPANY (US) 1981-01-20 US disclosed
US-4120856-A REACTING 3-HYDROXY-BENZODIAZEPINES WITH AMINOSULFUR TRIFLUORIDES E. I. DU PONT DE NEMOURS AND COMPANY (US) 1978-10-17 US disclosed