SCHEMBL11399663

SCHEMBL11399663

COc1cc2c(=O)c([S+](C)[O-])cn(C)c2cc1F

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TP53 P04637 3/20 0.34
NCOA1 Q15788 1/20 0.33
NCOA3 Q9Y6Q9 1/20 0.33
SMN1; SMN2 Q16637 2/20 0.32
KDM4E B2RXH2 1/20 0.32
GSK3B P49841 2/20 0.31
CDK1 P06493 1/20 0.31
CDK4 P11802 1/20 0.31
CCNB1 P14635 1/20 0.31
CCND1 P24385 1/20 0.31
CDK2 P24941 1/20 0.31
CDK5 Q00535 1/20 0.31
CDK5R1 Q15078 1/20 0.31
POLB P06746 2/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
LMNA P02545 1/20 0.31
THRB P10828 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11389627 0.89 TP53 (0.39) TP53SMN1; SMN2KDM4EGSK3BPOLB
SCHEMBL11398592 0.84 GSK3B (0.41) TP53SMN1; SMN2KDM4EGSK3BCDK1
SCHEMBL11402630 0.82 GSK3B (0.37) TP53SMN1; SMN2KDM4EGSK3BCDK1
SCHEMBL11401167 0.76 TP53 (0.34) TP53SMN1; SMN2POLBL3MBTL1THRB
SCHEMBL11391212 0.76 TP53 (0.36) TP53NCOA1NCOA3SMN1; SMN2GSK3B
SCHEMBL11399722 0.76 ADRB2 (0.47) KDM4EGSK3BPOLB
SCHEMBL11401796 0.76 ALDH1A1 (0.52) KDM4EGSK3BL3MBTL1
SCHEMBL11390014 0.75 ALDH1A1 (0.50) KDM4EGSK3BCDK1CCNB1CDK2
Flosequinan SCHEMBL122877 0.75 ATM (0.47) TP53KDM4EGSK3BCDK4CCND1
Flosequinan SCHEMBL5441172 0.75 ATM (0.47) TP53KDM4EGSK3BCDK4CCND1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4302460-A 4-Quinolinones having antihypertensive activity THE BOOTS COMPANY LIMITED (GB) 1981-11-24 US disclosed