SCHEMBL11401796

SCHEMBL11401796

COc1ccc2c(=O)c([S+](C)[O-])cn(C)c2c1

nearest known ligand 0.52

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.52
PTPN1 P18031 1/20 0.39
ADRB2 P07550 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.37
GSK3B P49841 4/20 0.37
PRKCA P17252 3/20 0.37
HTR6 P50406 1/20 0.36
NTRK1 P04629 2/20 0.36
KDM4E B2RXH2 2/20 0.36
MAPK1 P28482 1/20 0.36
HTT P42858 1/20 0.36
HSD17B10 Q99714 1/20 0.36
ABCG2 Q9UNQ0 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11399722 0.89 ADRB2 (0.47) ALDH1A1ADRB2GSK3BHTR6KDM4E
SCHEMBL9867248 0.85 MAT2A (0.39) ALDH1A1ADRB2HTR6KDM4E
SCHEMBL9868894 0.84 ALDH1A1 (0.36) ALDH1A1HTT
SCHEMBL11393569 0.83 PSEN1 (0.37) ALDH1A1L3MBTL1
SCHEMBL9869020 0.81 ALDH1A1 (0.37) ALDH1A1HTR6KDM4EMAPK1HTT
SCHEMBL7317623 0.81 TP53 (0.38) ALDH1A1GSK3BPRKCANTRK1KDM4E
Flosequinan SCHEMBL5441172 0.80 ATM (0.47) ALDH1A1GSK3BPRKCAKDM4E
Flosequinan SCHEMBL122877 0.80 ATM (0.47) ALDH1A1GSK3BPRKCAKDM4E
Flosequinan SCHEMBL5442796 0.80 ATM (0.47) ALDH1A1GSK3BPRKCAKDM4E
SCHEMBL10943341 0.80 NTRK1 (0.40) GSK3BNTRK1KDM4EMAPK1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4302460-A 4-Quinolinones having antihypertensive activity THE BOOTS COMPANY LIMITED (GB) 1981-11-24 US disclosed