SCHEMBL11399752

SCHEMBL11399752

C#CC=CC(Cc1cccc2ccccc12)NC

nearest known ligand 0.46

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 2/20 0.39
CTNNB1 P35222 1/20 0.38
CYP1A2 P05177 2/20 0.38
CYP2C19 P33261 2/20 0.38
CYP2D6 P10635 1/20 0.38
MTNR1A P48039 1/20 0.37
CYP2C9 P11712 1/20 0.37
ADRB2 P07550 4/20 0.36
MMP9 P14780 1/20 0.36
IFNAR1 P17181 1/20 0.35
NQO2 P16083 1/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7018449 0.81 SIGMAR1 (0.53) SIGMAR1CTNNB1CYP1A2CYP2C19CYP2D6
SCHEMBL9727662 0.79 CTNNB1 (0.45) SIGMAR1CTNNB1CYP1A2CYP2C19CYP2D6
SCHEMBL25660784 0.79 CTNNB1 (0.45) SIGMAR1CTNNB1CYP1A2CYP2C19CYP2D6
SCHEMBL9631575 0.79 CTNNB1 (0.45) SIGMAR1CTNNB1CYP1A2CYP2C19CYP2D6
SCHEMBL11397476 0.78 SIGMAR1 (0.37) SIGMAR1CTNNB1CYP1A2CYP2C19CYP2D6
SCHEMBL11407941 0.76 MME (0.36) SIGMAR1CTNNB1ADRB2MMP9
SCHEMBL9727658 0.70 CTNNB1 (0.45) SIGMAR1CTNNB1CYP1A2CYP2C19CYP2D6
SCHEMBL9631571 0.70 CTNNB1 (0.45) SIGMAR1CTNNB1CYP1A2CYP2C19CYP2D6
SCHEMBL31332073 0.69 NR3C1 (0.54) SIGMAR1CTNNB1CYP1A2CYP2C19CYP2D6
SCHEMBL16174128 0.69 NR3C1 (0.54) SIGMAR1CTNNB1CYP1A2CYP2C19CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0024587-A1 Propenylamines, processes for their production, pharmaceutical compositions containing them and their use as pharmaceuticals SANDOZ AG (CH) 1981-03-11 EP disclosed