SCHEMBL1144933

SCHEMBL1144933

Cc1cn([C@H]2CC[C@@H](CO)O2)c(=O)[nH]c1=S

nearest known ligand 0.59

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
TK1 P04183 5/20 0.59
LMNA P02545 4/20 0.45
ALB P02768 3/20 0.45
TSHR P16473 2/20 0.45
BLM P54132 2/20 0.45
PKM P14618 1/20 0.45
PMP22 Q01453 1/20 0.45
CYP2D6 P10635 1/20 0.45
ALDH1A1 P00352 2/20 0.44
MAPK1 P28482 1/20 0.44
POLB P06746 1/20 0.43
ADRA1A P35348 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14577794 1.00 TK1 (0.59) TK1LMNAALBTSHRBLM
SCHEMBL14421795 0.86 LMNA (0.58) TK1LMNAALBTSHRBLM
SCHEMBL925743 0.86 LMNA (0.58) TK1LMNAALBTSHRBLM
SCHEMBL29711774 0.86 LMNA (0.58) TK1LMNAALBTSHRBLM
SCHEMBL14596607 0.86 LMNA (0.58) TK1LMNAALBTSHRBLM
SCHEMBL23485 0.86 LMNA (0.58) TK1LMNAALBTSHRBLM
SCHEMBL762579 0.86 LMNA (0.58) TK1LMNAALBTSHRBLM
SCHEMBL13286394 0.86 LMNA (0.58) TK1LMNAALBTSHRBLM
SCHEMBL22992337 0.86 LMNA (0.58) TK1LMNAALBTSHRBLM
SCHEMBL27505365 0.86 LMNA (0.58) TK1LMNAALBTSHRBLM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 38 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2025024123-A1 NOVEL CITICOLINE DERIVATIVES THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2025-01-30 WO claimed
WO-2007083173-A2 MONONUCLEOTIDES AND MONONUCLEOSIDES FOR USE IN THERAPY UNIVERSITY OF DEBRECEN (HU) 2007-07-26 WO claimed
WO-1995011685-A1 2',3'-DIDEOXY-4'-THIORIBONUCLEOSIDES AS ANTIVIRAL AGENTS SOUTHERN RESEARCH INSTITUTE (US) 1995-05-04 WO claimed
US-20230037279-A9 METHOD FOR DIAGNOSING DISEASES USING MULTIPLEX FLUORESCENCE AND SEQUENCING MultiplexDX, s.r.o. (SK) 2023-02-02 US disclosed
US-20220002812-A1 METHOD FOR DIAGNOSING DISEASES USING MULTIPLEX FLUORESCENCE AND SEQUENCING MULTIPLEXDX S R O (SK) 2022-01-06 US disclosed
US-20210254067-A1 MICRORNA INHIBITORS FOR USE IN TREATING METABOLIC DISEASES HELMHOLTZ ZENTRUM MUENCHEN - DEUTSCHES FORSCHUNGSZENTRUM FUER GESUNDHEIT UND UMWELT (GMBH) (DE) 2021-08-19 US disclosed
EP-3850099-A1 MICRORNA INHIBITORS FOR USE IN TREATING METABOLIC DISEASES Helmholtz Zentrum München Forschungszentrum für Gesundheit und Umwelt GmbH (DE) 2021-07-21 EP disclosed
EP-3194597-B1 ALLELE-SPECIFIC THERAPY FOR HUNTINGTON DISEASE HAPLOTYPES UNIV BRITISH COLUMBIA (CA) 2021-06-30 EP disclosed
EP-3775277-A1 METHOD FOR DIAGNOSING DISEASES USING MULTIPLEX FLUORESCENCE AND SEQUENCING MultiplexDX, s.r.o. (SK) 2021-02-17 EP disclosed
US-10731160-B2 Allele-specific therapy for Huntington disease haplotypes THE UNIVERSITY OF BRITISH COLUMBIA (CA) 2020-08-04 US disclosed
US-20200199595-A1 ALLELE-SPECIFIC THERAPY FOR HUNTINGTON DISEASE HAPLOTYPES THE UNIVERSITY OF BRITISH COLUMBIA (CA) 2020-06-25 US disclosed
WO-2008106803-A1 DOUBLE-STRANDED LOCKED NUCLEIC ACID COMPOSITIONS NVENTA BIOPHARMACEUTICALS CORPORATION (US) 2008-09-12 WO disclosed
WO-2007083173-A2 MONONUCLEOTIDES AND MONONUCLEOSIDES FOR USE IN THERAPY UNIVERSITY OF DEBRECEN (HU) 2007-07-26 WO disclosed
EP-0974672-B1 Improved primers for AFLP amplification KEYGENE NV (NL) 2003-04-09 EP disclosed
US-6107039-A MIXING SAMPLE OF NUCLEIC ACID SEQUENCE TO BE ANALYZED WITH OLIGONUCLEOTIDE PROBE CONTAINING AT LEAST ONE THIOL-PROTECTED PYRIMIDINE NUCLEOTIDE, EXPOSING TO ENDONUCLEASE, AND IDENTIFYING FRAGMENTS HAVING HYBRIDIZED PROBE THE BOARD OF REGENTS OF THE UNIVERSITY OF OKLAHOMA 2000-08-22 US disclosed
EP-0974672-A1 Improved primers for AFLP amplification KEYGENE N.V. (NL) 2000-01-26 EP disclosed
US-6008334-A MODIFIED PYRIMIDINE NUCLEOSIDES/NUCLEOTIDES WITH PROTECTED THIOL GROUP ATTACHED AT 5 POSITION OF BASE THAT IS NOT INVOLVED IN WATSON-CRICK BASE PARING; FOR USE IN CHEMICAL AND ENZYMATIC SYNTHESIS OF NUCLEIC ACIDS THE BOARD OF REGENTS OF THE UNIVERSITY OF OKLAHOMA (US) 1999-12-28 US disclosed
WO-1998003532-A9 BASE-PROTECTED NUCLEOTIDE ANALOGS WITH PROTECTED THIOL GROUPS 1998-05-28 WO disclosed
WO-1995011685-A1 2',3'-DIDEOXY-4'-THIORIBONUCLEOSIDES AS ANTIVIRAL AGENTS SOUTHERN RESEARCH INSTITUTE (US) 1995-05-04 WO disclosed
US-4749647-A Polymerization-induced separation assay using recognition pairs GENETIC SYSTEMS CORPORATION (US) 1988-06-07 US disclosed