SCHEMBL1147672

SCHEMBL1147672

COc1ccc2nccc(OC[C@H]3CC[C@H](C(=O)Nc4ccc5c(c4)NC(=O)CS5)CC3)c2c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 2/20 0.48
KCNH2 Q12809 2/20 0.43
TP53 P04637 3/20 0.41
LMNA P02545 2/20 0.41
NPC1 O15118 2/20 0.41
POLB P06746 2/20 0.41
RAB9A P51151 2/20 0.41
HPGD P15428 1/20 0.41
TSHR P16473 1/20 0.41
NFKB1 P19838 1/20 0.41
HTT P42858 1/20 0.41
NFKB2 Q00653 1/20 0.41
RELA Q04206 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
GSK3B P49841 1/20 0.41
DDR2 Q16832 1/20 0.40
MAOA P21397 2/20 0.40
MAOB P27338 2/20 0.40
MTNR1A P48039 1/20 0.39
MTNR1B P49286 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3251532 0.89 MAOA (0.46) TRPV1KCNH2LMNADDR2MAOA
SCHEMBL1147911 0.89 TRPV1 (0.46) TRPV1KCNH2TP53LMNANPC1
SCHEMBL1147875 0.84 KCNH2 (0.47) TRPV1KCNH2MAOAMAOBMTNR1A
SCHEMBL1148106 0.82 SLC2A1 (0.51) TRPV1KCNH2
SCHEMBL1147944 0.82 SLC2A1 (0.51) TRPV1KCNH2
SCHEMBL1148032 0.82 SLC2A1 (0.51) TRPV1KCNH2
SCHEMBL1147533 0.79 KCNH2 (0.60) KCNH2TP53NPC1POLBRAB9A
SCHEMBL3256183 0.79 MAOA (0.46) TRPV1KCNH2LMNAMAOAMAOB
SCHEMBL1148044 0.78 TRPV1 (0.45) TRPV1KCNH2LMNAALDH1A1
SCHEMBL14341455 0.78 KCNH2 (0.65) KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7888359-B2 Cyclohexyl or piperidinyl carboxamide antibiotic derivatives ACTELION PHARMACEUTICAL LTD. (CH) 2011-02-15 US claimed
US-7888359-B2 Cyclohexyl or piperidinyl carboxamide antibiotic derivatives ACTELION PHARMACEUTICAL LTD. (CH) 2011-02-15 US disclosed