SCHEMBL3256183

SCHEMBL3256183

COc1ccc2ncnc(OCC3CCCCC3)c2c1.O=C(O)Nc1ccc2c(c1)NC(=O)CS2

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA P21397 2/20 0.46
MAOB P27338 2/20 0.46
PDGFRA P16234 3/20 0.41
KIT P10721 2/20 0.39
KDR P35968 2/20 0.38
MTNR1B P49286 3/20 0.38
MTNR1A P48039 1/20 0.38
BRAF P15056 1/20 0.38
MAPK14 Q16539 1/20 0.38
TNNI3K Q59H18 1/20 0.38
ALDH1A1 P00352 1/20 0.38
LMNA P02545 1/20 0.38
KCNH2 Q12809 1/20 0.38
PDE3B Q13370 1/20 0.37
PDE3A Q14432 1/20 0.37
EGFR P00533 1/20 0.37
MET P08581 1/20 0.37
CSF1R P07333 1/20 0.37
TRPV1 Q8NER1 1/20 0.37
ELANE P08246 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1147911 0.89 TRPV1 (0.46) MAOAMAOBKDRMTNR1BMTNR1A
SCHEMBL3251532 0.88 MAOA (0.46) MAOAMAOBPDGFRAKITALDH1A1
SCHEMBL3247108 0.80 MAPT (0.51) PDGFRAKITKDRMTNR1BMTNR1A
SCHEMBL1147672 0.79 TRPV1 (0.48) MAOAMAOBMTNR1BMTNR1AALDH1A1
SCHEMBL3252106 0.77 KCNH2 (0.46) MAOAMAOBMTNR1BMTNR1AALDH1A1
SCHEMBL3252103 0.73 KCNH2 (0.38) MAOAMAOBALDH1A1LMNAKCNH2
SCHEMBL3256206 0.72 MTNR1B (0.43) MAOAMAOBMTNR1BMTNR1AALDH1A1
SCHEMBL3249967 0.72 KCNH2 (0.45) KCNH2
SCHEMBL3251044 0.72 MTNR1B (0.53) MTNR1BMTNR1AALDH1A1LMNAEGFR
SCHEMBL3251040 0.72 MTNR1B (0.53) MTNR1BMTNR1AALDH1A1LMNAEGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2001478-B1 CYCLOHEXYL OR PIPERIDINYL CARBOXAMIDE ANTIBIOTIC DERIVATIVES ACTELION PHARMACEUTICALS LTD (CH) 2010-06-02 EP claimed