SCHEMBL11489482

SCHEMBL11489482

CC(O)(CCN1CCCC1)c1ccccc1-c1ccccc1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 6/20 0.50
CHRM2 P08172 5/20 0.50
CHRM1 P11229 5/20 0.50
KCNH2 Q12809 4/20 0.50
HTR1A P08908 3/20 0.50
OPRM1 P35372 3/20 0.50
LMNA P02545 2/20 0.50
MAPK1 P28482 2/20 0.46
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
CHRM3 P20309 4/20 0.44
KDM4E B2RXH2 4/20 0.44
CHRM4 P08173 3/20 0.44
CHRM5 P08912 3/20 0.44
SIGMAR1 Q99720 2/20 0.44
DRD2 P14416 1/20 0.44
DRD1 P21728 1/20 0.44
HTR2A P28223 1/20 0.44
DRD3 P35462 1/20 0.44
SCN1A P35498 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11487383 0.99 CYP2D6 (0.52) CYP2D6CHRM2CHRM1KCNH2HTR1A
SCHEMBL11492974 0.91 KDM4E (0.55) CYP2D6CHRM2CHRM1KCNH2HTR1A
SCHEMBL11487644 0.90 LMNA (0.49) CYP2D6CHRM2CHRM1KCNH2HTR1A
SCHEMBL11494400 0.90 CHRM4 (0.48) CHRM2CHRM1LMNAMEN1KMT2A
SCHEMBL11495151 0.89 KMT2A (0.49) LMNAMAPK1MEN1KMT2ACHRM3
SCHEMBL11492203 0.89 CHRM2 (0.47) CYP2D6CHRM2CHRM1KCNH2HTR1A
SCHEMBL11486718 0.88 KDM4E (0.48) OPRM1LMNAMEN1KMT2AKDM4E
SCHEMBL11489633 0.87 ALDH1A1 (0.52) LMNAMAPK1MEN1KMT2AKDM4E
SCHEMBL11488616 0.87 SLC6A4 (0.40) CYP2D6CHRM2CHRM1KCNH2HTR1A
SCHEMBL11487668 0.85 KDM4E (0.55) LMNAMEN1KMT2AKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4239759-A Morpholino containing compounds, compositions and use thereof MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1980-12-16 US disclosed
US-4110447-A Anti-inflammatory (halo-4-biphenylyl)-alkanolamines MERCK PATENT GESELLSCHAFT MIT BESCHRAENKTER HAFTUNG (DE) 1978-08-29 US disclosed