SCHEMBL11512880

SCHEMBL11512880

FC(F)(F)c1cccc(-c2cnn3cnnc3n2)c1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.53
ALDH1A1 P00352 2/20 0.53
LMNA P02545 1/20 0.46
IDO1 P14902 1/20 0.45
CTSS P25774 1/20 0.43
NOTUM Q6P988 1/20 0.42
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
GABRA1 P14867 1/20 0.41
HPGD P15428 1/20 0.41
GABRG2 P18507 1/20 0.41
GABRB3 P28472 1/20 0.41
GABRA5 P31644 1/20 0.41
GABRA3 P34903 1/20 0.41
GABRA2 P47869 1/20 0.41
HSD17B10 Q99714 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
ATR Q13535 1/20 0.41
AR P10275 1/20 0.41
KDM1A O60341 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11510818 0.79 KDM4E (0.47) KDM4EALDH1A1LMNAIDO1NOTUM
SCHEMBL11480435 0.77 KDM4E (0.57) KDM4EALDH1A1LMNAIDO1CTSS
SCHEMBL11514797 0.75 KDM4E (0.58) KDM4EALDH1A1LMNAIDO1CTSS
SCHEMBL11625891 0.73 ALDH1A1 (0.59) KDM4EALDH1A1LMNACYP1A2CYP3A4
SCHEMBL11512157 0.73 ALDH1A1 (0.43) KDM4EALDH1A1GABRG2GABRB3GABRA5
SCHEMBL3398455 0.71 ADORA2A (0.56) IDO1CTSSNOTUMCYP1A2CYP3A4
SCHEMBL9702800 0.70 KDM4E (0.62) KDM4EALDH1A1LMNAIDO1CTSS
SCHEMBL2463789 0.70 KDM4E (0.55) KDM4EALDH1A1LMNAIDO1CTSS
SCHEMBL11470852 0.69 MAOB (0.46) KDM4EALDH1A1NOTUMHSD17B10MAOB
SCHEMBL11478689 0.69 KDM4E (1.00) KDM4EALDH1A1LMNAIDO1CTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4159375-A 6- AND 7-Aryl-1,2,4-triazolo[4,3-b]-1,2,4-triazines AMERICAN CYANAMID COMPANY (US) 1979-06-26 US disclosed