SCHEMBL11519985

SCHEMBL11519985

C[Si](C)(C)c1ccccc1C(=O)NCC(=O)O

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 1/20 0.51
EGLN1 Q9GZT9 6/20 0.49
RAB9A P51151 1/20 0.49
GAA P10253 1/20 0.47
FTO Q9C0B1 3/20 0.47
BBOX1 O75936 1/20 0.47
KDM4C Q9H3R0 1/20 0.46
POLB P06746 2/20 0.46
EGLN2 Q96KS0 1/20 0.44
APEX1 P27695 1/20 0.43
KDM5B Q9UGL1 1/20 0.43
KDM2A Q9Y2K7 1/20 0.43
CYP2C19 P33261 1/20 0.43
KMT2A Q03164 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
KDM4E B2RXH2 1/20 0.42
MAPT P10636 1/20 0.42
HIF1A Q16665 1/20 0.42
SLC22A6 Q4U2R8 1/20 0.42
SLC22A8 Q8TCC7 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7219605 0.84 L3MBTL1 (0.49) KMT2ATSHRHTT
SCHEMBL31448014 0.83 KEAP1 (0.62) KEAP1EGLN1RAB9AGAAFTO
SCHEMBL1285567 0.79 HPGD (0.62) KEAP1RAB9AGAACYP2C19KMT2A
SCHEMBL30319510 0.79 HPGD (0.62) KEAP1RAB9AGAACYP2C19KMT2A
SCHEMBL7738430 0.78 GAA (0.55) GAAPOLB
SCHEMBL27450922 0.78 KEAP1 (0.66) KEAP1EGLN1RAB9AGAAFTO
SCHEMBL30289977 0.78 KMT2A (0.65) KEAP1EGLN1KDM4CAPEX1CYP2C19
SCHEMBL6844310 0.77 KEAP1 (0.53) KEAP1EGLN1RAB9AGAAKMT2A
SCHEMBL8116346 0.77 HPGD (0.60) KEAP1RAB9AGAACYP2C19KMT2A
Salicyluric Acid SCHEMBL570541 0.77 HPGD (0.58) KEAP1EGLN1RAB9AGAAFTO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4162319-A ANTHELMINTICS, PSYCHOTROPIC, CNS, HYPOGLYCOMIC AGENTS MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1979-07-24 US disclosed
US-4120961-A ANTIHELMINTICS, CNS ACITVITY E. MERCK (DE) 1978-10-17 US disclosed
US-4051243-A RING SUBSTITUTED PYRAZINO-ISOQUINOLINE DERIVATIVES AND THEIR PREPARATION MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DT) 1977-09-27 US disclosed