SCHEMBL11520974

SCHEMBL11520974

O=C(NC(=O)c1c(Cl)cccc1Cl)Nc1cnc(C2CCCC2)cn1

nearest known ligand 0.45

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TYK2 P29597 6/20 0.45
JAK2 O60674 5/20 0.45
JAK1 P23458 2/20 0.42
CDK9 P50750 1/20 0.41
JAK3 P52333 1/20 0.41
ABL1 P00519 1/20 0.41
TAS1R3 Q7RTX0 2/20 0.41
TAS1R1 Q7RTX1 2/20 0.41
TAS1R2 Q8TE23 2/20 0.41
PPIA P62937 1/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
PDE10A Q9Y233 1/20 0.39
MAPT P10636 2/20 0.39
MAPK14 Q16539 1/20 0.38
ATR Q13535 1/20 0.38
HCRTR1 O43613 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11521457 0.95 JAK2 (0.43) TYK2JAK2JAK1CDK9JAK3
SCHEMBL11524573 0.80 RAB9A (0.46) TYK2JAK2JAK1CDK9JAK3
SCHEMBL11519411 0.80 RAB9A (0.47) TYK2JAK2JAK1PPIANPC1
SCHEMBL11526196 0.79 JAK2 (0.41) TYK2JAK2JAK1CDK9JAK3
SCHEMBL11522976 0.78 RAB9A (0.45) TYK2JAK2JAK1PPIANPC1
SCHEMBL11525516 0.77 PPIA (0.48) TYK2JAK2JAK1ABL1PPIA
SCHEMBL11604630 0.77 RAB9A (0.48) TYK2JAK2PPIANPC1RAB9A
SCHEMBL11521949 0.77 ABL1 (0.43) TYK2JAK2JAK1CDK9JAK3
SCHEMBL11385328 0.76 RAB9A (0.47) TYK2JAK2JAK1PPIANPC1
SCHEMBL11521149 0.75 NPC1 (0.46) TYK2JAK2PPIANPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4160834-A INSECTICIDES ELI LILLY AND COMPANY (US) 1979-07-10 US disclosed
US-4083977-A Novel insecticidal 1-(substituted benzoyl)-3-(substituted pyrazinyl)ureas ELI LILLY AND COMPANY (US) 1978-04-11 US disclosed