SCHEMBL11522976

SCHEMBL11522976

O=C(NC(=O)c1c(Cl)cccc1Cl)Nc1cnc(Br)cn1

nearest known ligand 0.45

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 3/20 0.45
NPC1 O15118 1/20 0.45
PPIA P62937 1/20 0.42
HDAC1 Q13547 1/20 0.41
TYK2 P29597 8/20 0.41
JAK2 O60674 7/20 0.41
JAK1 P23458 4/20 0.41
CYP3A4 P08684 1/20 0.41
KDM4E B2RXH2 2/20 0.40
MAPT P10636 3/20 0.40
GHSR Q92847 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11519411 0.86 RAB9A (0.47) RAB9ANPC1PPIATYK2JAK2
SCHEMBL8656115 0.84 RAB9A (0.56) RAB9ANPC1KDM4EMAPT
SCHEMBL11524573 0.84 RAB9A (0.46) RAB9ANPC1PPIATYK2JAK2
SCHEMBL11519534 0.83 RAB9A (0.40) RAB9ANPC1PPIAHDAC1TYK2
SCHEMBL11524038 0.81 RAB9A (0.41) RAB9ANPC1PPIAHDAC1TYK2
SCHEMBL11163699 0.81 RAB9A (0.68) RAB9ANPC1MAPT
SCHEMBL11604630 0.81 RAB9A (0.48) RAB9ANPC1PPIATYK2JAK2
SCHEMBL11523665 0.81 HCRTR1 (0.48) RAB9ANPC1TYK2KDM4EMAPT
SCHEMBL11525363 0.81 CHEK1 (0.54)
SCHEMBL11519925 0.81 TYK2 (0.46) RAB9ANPC1PPIAHDAC1TYK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4160834-A INSECTICIDES ELI LILLY AND COMPANY (US) 1979-07-10 US claimed
US-4160834-A INSECTICIDES ELI LILLY AND COMPANY (US) 1979-07-10 US disclosed
US-4083977-A Novel insecticidal 1-(substituted benzoyl)-3-(substituted pyrazinyl)ureas ELI LILLY AND COMPANY (US) 1978-04-11 US disclosed