SCHEMBL11530516

SCHEMBL11530516

Clc1cc2c(cc1Cl)Nc1cscc1C(N1CCNCC1)=N2

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 8/20 0.51
CHRM1 P11229 6/20 0.51
CHRM2 P08172 4/20 0.51
CHRM4 P08173 4/20 0.51
CHRM5 P08912 4/20 0.51
CHRM3 P20309 4/20 0.51
DRD1 P21728 4/20 0.51
KCNH2 Q12809 4/20 0.51
CYP1A2 P05177 3/20 0.51
CYP3A4 P08684 3/20 0.51
CYP2D6 P10635 3/20 0.51
MTOR P42345 2/20 0.51
ADRA2A P08913 4/20 0.41
HTR2A P28223 4/20 0.41
HRH1 P35367 4/20 0.41
ADRA2B P18089 3/20 0.41
ADRA2C P18825 3/20 0.41
ADRA1D P25100 3/20 0.41
HTR2C P28335 3/20 0.41
ADRA1A P35348 3/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11534075 0.86 CHRM1 (0.52) DRD2CHRM1CHRM2CHRM4CHRM5
SCHEMBL11528346 0.85 DRD2 (0.71) DRD2CHRM1CHRM2CHRM4CHRM5
SCHEMBL3407124 0.81 DRD2 (0.76) DRD2CHRM1CHRM2CHRM4CHRM5
SCHEMBL11529615 0.81 CHRM1 (0.57) DRD2CHRM1CHRM2CHRM4CHRM5
SCHEMBL11535575 0.80 DRD2 (0.60) DRD2CHRM1CHRM2CHRM4CHRM5
SCHEMBL11531463 0.78 HRH4 (0.44) DRD2CHRM1CHRM2CHRM4CHRM5
SCHEMBL11531459 0.78 DRD2 (0.36) DRD2CHRM1CHRM2CHRM4CHRM5
SCHEMBL11634458 0.78 DRD2 (0.46) DRD2CHRM1CHRM2CHRM4CHRM5
SCHEMBL11635354 0.78 DRD2 (0.43) DRD2CHRM1CHRM2CHRM4CHRM5
SCHEMBL11629502 0.77 DRD2 (0.44) DRD2CHRM1CHRM2CHRM4CHRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4172831-A CENTRAL NERVOUS SYSTEM LILLY INDUSTRIES LIMITED (GB) 1979-10-30 US disclosed
US-4115574-A CNS ACTIVITY LILLY INDUSTRIES LIMITED (GB) 1978-09-19 US disclosed
US-4115568-A CNS ACTIVITY LILLY INDUSTRIES LIMITED (GB) 1978-09-19 US disclosed