SCHEMBL11529615

SCHEMBL11529615

Fc1ccc2c(c1)N=C(N1CCNCC1)c1cscc1N2

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM1 P11229 3/20 0.57
HRH1 P35367 2/20 0.57
PAK1 Q13153 1/20 0.57
DRD2 P14416 3/20 0.52
CHRM2 P08172 2/20 0.52
CHRM4 P08173 2/20 0.52
CHRM5 P08912 2/20 0.52
CHRM3 P20309 2/20 0.52
DRD1 P21728 2/20 0.52
KCNH2 Q12809 2/20 0.52
CYP1A2 P05177 1/20 0.52
CYP3A4 P08684 1/20 0.52
CYP2D6 P10635 1/20 0.52
MTOR P42345 1/20 0.52
ADRA2A P08913 1/20 0.45
ADRA2B P18089 1/20 0.45
ADRA2C P18825 1/20 0.45
ADRA1D P25100 1/20 0.45
HTR2A P28223 1/20 0.45
HTR2C P28335 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11530673 0.87 CHRM1 (0.76) CHRM1HRH1PAK1
SCHEMBL11528346 0.86 DRD2 (0.71) CHRM1HRH1DRD2CHRM2CHRM4
SCHEMBL3414200 0.83 CHRM1 (0.74) CHRM1HRH1PAK1DRD2CHRM2
SCHEMBL11535575 0.83 DRD2 (0.60) CHRM1HRH1DRD2CHRM2CHRM4
SCHEMBL11536340 0.82 CHRM1 (0.56) CHRM1HRH1PAK1
SCHEMBL11530516 0.81 DRD2 (0.51) CHRM1HRH1PAK1DRD2CHRM2
SCHEMBL3429232 0.79 CHRM1 (0.68) CHRM1HRH1PAK1DRD2CHRM2
SCHEMBL3410996 0.79 DRD2 (0.74) CHRM1HRH1PAK1DRD2CHRM2
SCHEMBL11531624 0.79 CHRM1 (0.54) CHRM1HRH1PAK1DRD2CHRM2
SCHEMBL11531571 0.78 CHRM1 (0.52) CHRM1HRH1PAK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4172831-A CENTRAL NERVOUS SYSTEM LILLY INDUSTRIES LIMITED (GB) 1979-10-30 US disclosed
US-4115568-A CNS ACTIVITY LILLY INDUSTRIES LIMITED (GB) 1978-09-19 US disclosed
US-4115574-A CNS ACTIVITY LILLY INDUSTRIES LIMITED (GB) 1978-09-19 US disclosed