SCHEMBL11530807

SCHEMBL11530807

Cc1ccc(/C=C/c2ccc(I)cc2)cc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NFE2L2 Q16236 6/20 0.58
APP P05067 1/20 0.58
RELA Q04206 1/20 0.54
PTGS1 P23219 2/20 0.50
PTGS2 P35354 2/20 0.50
ALOX5 P09917 1/20 0.50
CA1 P00915 1/20 0.48
CYP2A6 P11509 1/20 0.46
TUBB4A P04350 1/20 0.45
TUBB P07437 1/20 0.45
TUBA3C P0DPH7 1/20 0.45
TUBA1B P68363 1/20 0.45
TUBA4A P68366 1/20 0.45
TUBB4B P68371 1/20 0.45
TUBB3 Q13509 1/20 0.45
TUBB2A Q13885 1/20 0.45
TUBB8 Q3ZCM7 1/20 0.45
TUBA3E Q6PEY2 1/20 0.45
TUBA1A Q71U36 1/20 0.45
TUBA1C Q9BQE3 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11530814 1.00 NFE2L2 (0.58) NFE2L2APPRELAPTGS1PTGS2
SCHEMBL5617807 0.87 APP (0.62) NFE2L2APPRELAPTGS1PTGS2
SCHEMBL17311315 0.87 APP (0.62) NFE2L2APPRELAPTGS1PTGS2
SCHEMBL699783 0.86 APP (0.64) NFE2L2APPPTGS1CA1
SCHEMBL699782 0.86 APP (0.64) NFE2L2APPPTGS1CA1
(E)-1,2-Di-P-Tolylethene SCHEMBL1793692 0.86 NFE2L2 (0.74) NFE2L2RELAPTGS1PTGS2ALOX5
SCHEMBL318786 0.86 NFE2L2 (0.74) NFE2L2RELAPTGS1PTGS2ALOX5
(E)-1,2-Di-P-Tolylethene SCHEMBL1305582 0.86 NFE2L2 (0.74) NFE2L2RELAPTGS1PTGS2ALOX5
(E)-1,2-Di-P-Tolylethene SCHEMBL1305580 0.86 NFE2L2 (0.74) NFE2L2RELAPTGS1PTGS2ALOX5
SCHEMBL318785 0.86 NFE2L2 (0.74) NFE2L2RELAPTGS1PTGS2ALOX5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2968440-B1 CYTOTOXIC AND ANTI-MITOTIC COMPOUNDS, AND METHODS OF USING THE SAME ZYMEWORKS INC (CA) 2019-06-05 EP disclosed
US-4153719-A Aromatic diketones STERLING DRUG INC. (US) 1979-05-08 US disclosed