SCHEMBL11533443

SCHEMBL11533443

N#CCOC(=O)c1ccc(C(c2ccccc2)(c2cccc(F)c2)c2cccc(F)c2)cn1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNN4 O15554 4/20 0.36
ALDH1A1 P00352 2/20 0.34
ALOX15 P16050 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
HSD17B10 Q99714 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
HDAC3 O15379 1/20 0.34
HDAC1 Q13547 1/20 0.34
HDAC2 Q92769 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34
MAPK1 P28482 1/20 0.34
GABRA1 P14867 2/20 0.33
GABRG2 P18507 2/20 0.33
GABRB3 P28472 2/20 0.33
GABRA5 P31644 2/20 0.33
GABRA3 P34903 2/20 0.33
GABRA2 P47869 2/20 0.33
GRM5 P41594 2/20 0.33
GABRA4 P48169 1/20 0.33
GABRA6 Q16445 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11533431 0.97 HDAC3 (0.35) KCNN4ALDH1A1ALOX15NPSR1HSD17B10
SCHEMBL11534104 0.91 MAPT (0.36) KCNN4ALDH1A1ALOX15NPSR1HSD17B10
SCHEMBL11534109 0.90 ALDH1A1 (0.38) ALDH1A1L3MBTL1GABRA1GABRG2GABRB3
SCHEMBL11542791 0.87 MEN1 (0.39) ALDH1A1L3MBTL1MAPK1GABRA1GABRG2
SCHEMBL11534846 0.87 ALDH1A1 (0.39) ALDH1A1GABRA1GABRG2GABRB3GABRA5
SCHEMBL11536526 0.87 KMT2A (0.41) ALDH1A1L3MBTL1MAPK1GABRA1GABRG2
SCHEMBL11541337 0.87 MAPK1 (0.43) ALDH1A1ALOX15L3MBTL1MAPK1GABRA1
SCHEMBL11538505 0.85 GABRA1 (0.40) ALDH1A1ALOX15HSD17B10GABRA1GABRG2
SCHEMBL11536196 0.84 ALDH1A1 (0.39) ALDH1A1L3MBTL1GABRA1GABRG2GABRB3
SCHEMBL11536777 0.84 ALDH1A1 (0.39) ALDH1A1GABRA1GABRG2GABRB3GABRA5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4139625-A 5-(Substituted triphenylmethyl)picolinamides and their use as anti-acne agents SCHERING CORPORATION (US) 1979-02-13 US disclosed
US-4133887-A Trityl picolinic acid derivatives and their use as anti-acne agents SCHERING CORPORATION (US) 1979-01-09 US disclosed
US-4127662-A ANTIACNE SCHERING CORPORATION (US) 1978-11-28 US disclosed
US-4123433-A ANTIACNE AGENTS SCHERING CORPORATION (US) 1978-10-31 US disclosed
US-4044140-A Trityl picolinic acid derivatives and their use as anti-acne agents SCHERING CORPORATION (US) 1977-08-23 US disclosed