SCHEMBL11533786

SCHEMBL11533786

O=C1NC(=O)C(c2cccnc2)N1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.50
CHRNB2 P17787 5/20 0.47
CHRNA4 P43681 5/20 0.47
CYP2A6 P11509 3/20 0.47
MAPK1 P28482 2/20 0.46
GAA P10253 1/20 0.46
RAB9A P51151 1/20 0.44
CHRNA7 P36544 4/20 0.44
CYP11B2 P19099 1/20 0.43
HTT P42858 1/20 0.43
MEN1 O00255 3/20 0.42
KMT2A Q03164 3/20 0.42
CYP2D6 P10635 2/20 0.42
CYP2C19 P33261 2/20 0.42
POLB P06746 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP2C9 P11712 1/20 0.42
KDM4E B2RXH2 2/20 0.42
TSHR P16473 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17622810 0.78 TDP1 (0.61) TDP1GAARAB9AHTTSMN1; SMN2
SCHEMBL19955179 0.77 TDP1 (0.66) TDP1GAAHTTKMT2APOLB
SCHEMBL31738422 0.77 TDP1 (0.66) TDP1GAAHTTKMT2APOLB
SCHEMBL395878 0.77 TDP1 (0.66) TDP1GAAHTTKMT2APOLB
SCHEMBL13527924 0.75 TDP1 (0.80) TDP1GAAMEN1KMT2AKDM4E
SCHEMBL8234663 0.75 TDP1 (0.53) TDP1GAAKDM4ETSHRALDH1A1
SCHEMBL10242198 0.74 CHRNB2 (0.53) CHRNB2CHRNA4CYP2A6MAPK1GAA
SCHEMBL156842 0.73 CHRNB2 (0.56) TDP1CHRNB2CHRNA4CYP2A6MAPK1
SCHEMBL10146593 0.72 ALDH1A1 (0.74) TDP1MAPK1GAACYP11B2MEN1
SCHEMBL10375118 0.72 CHRNB2 (0.56) CHRNB2CHRNA4CYP2A6MAPK1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016044777-A1 HAT INHIBITORS AND METHODS FOR THEIR USE ABBVIE INC. (US) 2016-03-24 WO disclosed
WO-2010054279-A1 COMPOUNDS FOR THE TREATMENT OF INFLAMMATORY DISORDERS SCHERING CORPORATION (US) 2010-05-14 WO disclosed
US-4179511-A Antibacterial 3-(5-tetrazolyl) penam compounds PFIZER INC. (US) 1979-12-18 US disclosed
US-4143039-A ANTIBACTERIAL 3-(5-TETRAZOLYL)PENAM COMPOUNDS PFIZER INC. (US) 1979-03-06 US disclosed
US-4115385-A PENICILLINS PFIZER INC. (US) 1978-09-19 US disclosed