SCHEMBL11534209

SCHEMBL11534209

Cc1ccc2c(c1)C(=O)C1(CC1)N2

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.47
KDM4E B2RXH2 4/20 0.47
MAPT P10636 3/20 0.47
HPGD P15428 1/20 0.47
HSD17B10 Q99714 1/20 0.47
ROS1 P08922 1/20 0.46
CDK5 Q00535 1/20 0.46
ACVR1 Q04771 1/20 0.46
LRRK2 Q5S007 1/20 0.46
EPHX2 P34913 1/20 0.46
CA1 P00915 2/20 0.43
CA2 P00918 2/20 0.43
CA4 P22748 2/20 0.43
CA7 P43166 2/20 0.43
CA9 Q16790 2/20 0.43
GAA P10253 1/20 0.41
CSNK1G1 Q9HCP0 1/20 0.40
METAP1 P53582 1/20 0.40
CYP1A2 P05177 1/20 0.39
POLB P06746 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16170237 0.93 POLB (0.45) ALDH1A1KDM4EMAPTHPGDHSD17B10
SCHEMBL11538334 0.80 CES1 (0.53) MAPTLRRK2
SCHEMBL11539506 0.80 ALDH1A1 (0.57) ALDH1A1KDM4EMAPTHPGDLRRK2
SCHEMBL16170247 0.79 ALDH1A1 (0.53) ALDH1A1KDM4EMAPTHPGDHSD17B10
SCHEMBL11536434 0.75 MAOA (0.47) ALDH1A1KDM4EHPGDHSD17B10ACVR1
SCHEMBL24649691 0.74 CYP1A2 (0.46) ALDH1A1KDM4EMAPTHPGDHSD17B10
SCHEMBL16170250 0.74 KDM4E (0.47) ALDH1A1KDM4EMAPTHPGDHSD17B10
SCHEMBL15219327 0.74 ROS1 (0.54) ALDH1A1KDM4EMAPTHPGDHSD17B10
SCHEMBL16163174 0.74 PDE7A (0.62) ALDH1A1KDM4EMAPTHPGDHSD17B10
SCHEMBL16170245 0.73 ALDH1A1 (0.46) ALDH1A1KDM4EMAPTHPGDHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4154731-A ANTISECRETORY AGENTS, ANTIINFLAMMATORY AGENTS, ANALGESICS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1979-05-15 US disclosed
US-4105670-A ANTISECRETORY, ANTIINFLAMMATORY, ANALGESIC, DECARBOXYLATION TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1978-08-08 US disclosed