SCHEMBL11534252

SCHEMBL11534252

Cc1c(C(=O)c2cccs2)cc2cc(C(=O)O)oc2c1C

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 5/20 0.48
RAB9A P51151 4/20 0.48
ALOX15 P16050 3/20 0.48
MAPT P10636 3/20 0.48
MAPK1 P28482 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
NPSR1 Q6W5P4 1/20 0.48
LMNA P02545 1/20 0.48
ALDH1A1 P00352 3/20 0.45
HSD17B10 Q99714 2/20 0.45
PSMD14 O00487 1/20 0.45
MMP2 P08253 1/20 0.45
DAO P14920 1/20 0.41
HPGDS O60760 1/20 0.41
GPR35 Q9HC97 2/20 0.40
ADORA1 P30542 2/20 0.40
ADORA2A P29274 1/20 0.40
HPGD P15428 4/20 0.39
MEN1 O00255 3/20 0.39
KMT2A Q03164 3/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11535276 0.89 NPC1 (0.45) NPC1RAB9AALOX15MAPTMAPK1
SCHEMBL11532310 0.82 MAPT (0.48) NPC1RAB9AALOX15MAPTMAPK1
SCHEMBL11535872 0.81 NPC1 (0.53) NPC1RAB9AALOX15MAPTMAPK1
SCHEMBL11535994 0.76 MAPT (0.53) NPC1RAB9AALOX15MAPTMAPK1
SCHEMBL11530620 0.71 MAPT (0.44) NPC1RAB9AALOX15MAPTMAPK1
SCHEMBL5772064 0.70 PIM1 (0.46) LMNADAOGPR35KMT2AKDM4E
SCHEMBL11825410 0.69 GPR35 (0.43) ALDH1A1GPR35
SCHEMBL11834711 0.68 GPR35 (0.42) ALOX15MAPTLMNAALDH1A1HSD17B10
SCHEMBL6292875 0.67 MCL1 (0.49) MAPTSMN1; SMN2LMNAALDH1A1HSD17B10
SCHEMBL3859942 0.66 ALOX15 (1.00) NPC1RAB9AALOX15MAPTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4085117-A DIURETIC-SALURETIC, URICOSURIC, HYPOTENSIVE, ANTIKALURETIC AGENTS MERCK & CO., INC. (US) 1978-04-18 US claimed
US-4154742-A DIURETICS MERCK & CO., INC. (US) 1979-05-15 US disclosed
US-4085117-A DIURETIC-SALURETIC, URICOSURIC, HYPOTENSIVE, ANTIKALURETIC AGENTS MERCK & CO., INC. (US) 1978-04-18 US disclosed