SCHEMBL11535191

SCHEMBL11535191

Cc1cccc(C(=O)c2ccc3n2CCC3C#N)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDC42 P60953 3/20 0.47
RAC1 P63000 3/20 0.47
PTGS2 P35354 3/20 0.47
PTGS1 P23219 2/20 0.47
NPC1 O15118 2/20 0.47
RAB9A P51151 2/20 0.47
CHRM3 P20309 1/20 0.47
OPRM1 P35372 1/20 0.47
PAK1 Q13153 1/20 0.47
ABCC4 O15439 1/20 0.40
HTT P42858 1/20 0.40
BLM P54132 1/20 0.40
LMNA P02545 1/20 0.40
CYP1A2 P05177 1/20 0.40
NFKB1 P19838 1/20 0.40
MAPK1 P28482 1/20 0.40
HPGD P15428 1/20 0.39
HSD11B1 P28845 1/20 0.39
MGLL Q99685 1/20 0.39
CYP2C19 P33261 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11350964 0.86 CDC42 (0.47) CDC42RAC1PTGS2PTGS1NPC1
SCHEMBL11340159 0.86 CDC42 (0.47) CDC42RAC1PTGS2PTGS1NPC1
SCHEMBL11533036 0.85 PTGS2 (0.48) CDC42RAC1PTGS2PTGS1NPC1
SCHEMBL7905025 0.85 PTGS2 (0.64) CDC42RAC1PTGS2PTGS1NPC1
SCHEMBL11444567 0.84 CDC42 (0.44) CDC42RAC1PTGS2PTGS1NPC1
SCHEMBL20121862 0.83 CDC42 (0.51) CDC42RAC1PTGS2PTGS1NPC1
SCHEMBL11437849 0.82 CDC42 (0.42) CDC42RAC1PTGS2PTGS1NPC1
SCHEMBL10961188 0.81 PTGS2 (0.74) CDC42RAC1PTGS2PTGS1NPC1
SCHEMBL11438541 0.80 CDC42 (0.40) CDC42RAC1PTGS2PTGS1NPC1
SCHEMBL11202947 0.79 FAAH (0.41) NPC1RAB9AMAPK1HPGDHSD11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4140698-A 1,2-Dihydro-3H-pyrrolo[1,2-a]pyrrole-1-nitriles SYNTEX (USA) INC. (US) 1979-02-20 US disclosed
EP-0000649-A1 5-substituted-1,2-dihydro-3H-pyrrolo(1,2-a)pyrrole-1-carbonitriles and process for their conversion to the corresponding 1-carboxylic acids SYNTEX (U.S.A.) INC. (US) 1979-02-07 EP disclosed