SCHEMBL11536103

SCHEMBL11536103

Fc1cccc(C(c2ccc(Br)nc2)(c2cccc(F)c2)c2cccc(F)c2)c1

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 2/20 0.42
KCNN4 O15554 4/20 0.39
HDAC6 Q9UBN7 2/20 0.38
HDAC3 O15379 1/20 0.38
HDAC1 Q13547 1/20 0.38
HDAC2 Q92769 1/20 0.38
PTPN1 P18031 1/20 0.33
KIF11 P52732 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
USP2 O75604 1/20 0.32
KMT2A Q03164 1/20 0.32
ACHE P22303 1/20 0.31
MAOB P27338 1/20 0.31
MAP4K4 O95819 1/20 0.31
NFE2L2 Q16236 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11537554 0.95 KCNN4 (0.40) CYP19A1KCNN4HDAC6HDAC3HDAC1
SCHEMBL11536641 0.85 MAPK1 (0.39) CYP19A1HDAC6HDAC3HDAC1HDAC2
SCHEMBL11535231 0.83 KCNN4 (0.39) CYP19A1KCNN4KIF11TDP1USP2
SCHEMBL11533304 0.80 KIF11 (0.38) KIF11TDP1KMT2AMAOB
SCHEMBL11534894 0.80 NPC1 (0.33) CYP19A1KCNN4
SCHEMBL11554435 0.78 DGAT1 (0.39) CYP19A1KCNN4KMT2AMAP4K4
SCHEMBL11534919 0.76 KMO (0.47) CYP19A1KCNN4HDAC6HDAC3HDAC1
SCHEMBL11541379 0.76 ALDH1A1 (0.48) CYP19A1KIF11TDP1KMT2A
SCHEMBL11535667 0.75 KIF11 (0.40) KIF11KMT2A
SCHEMBL11535031 0.74 KCNN4 (0.46) CYP19A1KCNN4HDAC6HDAC3HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4139625-A 5-(Substituted triphenylmethyl)picolinamides and their use as anti-acne agents SCHERING CORPORATION (US) 1979-02-13 US disclosed
US-4133887-A Trityl picolinic acid derivatives and their use as anti-acne agents SCHERING CORPORATION (US) 1979-01-09 US disclosed
US-4127662-A ANTIACNE SCHERING CORPORATION (US) 1978-11-28 US disclosed
US-4123433-A ANTIACNE AGENTS SCHERING CORPORATION (US) 1978-10-31 US disclosed
US-4044140-A Trityl picolinic acid derivatives and their use as anti-acne agents SCHERING CORPORATION (US) 1977-08-23 US disclosed