SCHEMBL11535398

SCHEMBL11535398

O=c1[nH]cc(C(c2ccc(F)cc2)c2ccc(F)cc2)cc1C(c1ccc(F)cc1)c1ccc(F)cc1

nearest known ligand 0.42

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.42
POLB P06746 1/20 0.42
ERCC1 P07992 1/20 0.40
ERCC4 Q92889 1/20 0.40
DAO P14920 5/20 0.37
PTGDR2 Q9Y5Y4 1/20 0.35
AKR1C3 P42330 1/20 0.35
EPHX2 P34913 1/20 0.33
MAPT P10636 1/20 0.33
MAPK14 Q16539 1/20 0.32
CYP19A1 P11511 1/20 0.32
CYP11B1 P15538 1/20 0.32
CYP11B2 P19099 1/20 0.32
KDM4E B2RXH2 1/20 0.32
ROCK2 O75116 1/20 0.32
MET P08581 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11536497 0.83 CYP19A1 (0.40) DAOCYP19A1
SCHEMBL11542166 0.83 GAA (0.45) GAADAOMAPT
SCHEMBL11540707 0.82 DAO (0.39) DAOMAPTKDM4E
SCHEMBL3165240 0.78 EPHX2 (0.46) GAAPOLBERCC1ERCC4DAO
SCHEMBL11538902 0.70 ACP3 (0.39) GAADAOMAPTKDM4EROCK2
SCHEMBL2489611 0.69 IDO1 (0.50) GAAPOLBCYP19A1
SCHEMBL11537810 0.69 NR3C1 (0.44) GAAMAPTCYP19A1CYP11B1CYP11B2
SCHEMBL30821590 0.68 IDO1 (0.39) GAAPOLBCYP19A1CYP11B1CYP11B2
SCHEMBL31005301 0.64 CYP19A1 (0.36) GAACYP19A1CYP11B1CYP11B2
SCHEMBL11537244 0.63 BRD4 (0.43) DAOMAPTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4138488-A Diphenylmethyl picolinic acid derivatives and their use as anti-acne agents SCHERING CORPORATION (US) 1979-02-06 US disclosed