SCHEMBL11543010

SCHEMBL11543010

CC(=O)Oc1cc(=O)n(-c2ccccc2Br)c2ccccc12

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.42
NPSR1 Q6W5P4 1/20 0.40
PTPN1 P18031 1/20 0.40
PTGS2 P35354 1/20 0.40
ALDH1A1 P00352 4/20 0.39
RECQL P46063 1/20 0.39
HSD17B10 Q99714 1/20 0.39
MAPT P10636 1/20 0.38
PKM P14618 1/20 0.38
APLNR P35414 1/20 0.38
BRD4 O60885 1/20 0.38
SHMT2 P34897 1/20 0.38
TSHR P16473 2/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
SLC22A6 Q4U2R8 1/20 0.37
KDM4E B2RXH2 1/20 0.36
POLB P06746 1/20 0.36
GSK3A P49840 1/20 0.36
GSK3B P49841 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11541711 0.86 MAPT (0.47) HTTNPSR1PTPN1PTGS2ALDH1A1
SCHEMBL11542874 0.85 PTPN1 (0.42) HTTNPSR1PTPN1PTGS2ALDH1A1
SCHEMBL11540561 0.85 TSHR (0.45) HTTALDH1A1RECQLHSD17B10APLNR
SCHEMBL11540070 0.82 NPSR1 (0.46) HTTNPSR1PTPN1PTGS2ALDH1A1
SCHEMBL11541058 0.81 ALDH1A1 (0.42) HTTPTPN1PTGS2ALDH1A1RECQL
SCHEMBL11540274 0.81 NPSR1 (0.47) HTTNPSR1PTPN1PTGS2ALDH1A1
SCHEMBL11575819 0.80 HTT (0.40) HTTNPSR1PTPN1PTGS2ALDH1A1
SCHEMBL11542615 0.77 NPSR1 (0.46) HTTNPSR1PTPN1PTGS2BRD4
SCHEMBL11541055 0.77 NPSR1 (0.46) HTTNPSR1PTPN1ALDH1A1HSD17B10
SCHEMBL29206051 0.76 KCNA3 (0.56) ALDH1A1HSD17B10BRD4TSHRSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4168312-A Quinolone derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1979-09-18 US disclosed