SCHEMBL11544650

SCHEMBL11544650

O=C1C=C2CCN(CCc3ccccc3)CC(c3ccccc3)C2=CC1=O

nearest known ligand 0.47

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 4/20 0.44
SLC6A3 Q01959 1/20 0.41
GRIN1 Q05586 2/20 0.40
GRIN2B Q13224 2/20 0.40
ACHE P22303 1/20 0.40
DRD2 P14416 1/20 0.39
DRD3 P35462 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11549587 0.89 TACR1 (0.46) SIGMAR1GRIN1GRIN2B
Bromide SCHEMBL11478757 0.85 SLC18A3 (0.43) DRD2
Hydrochloric Acid SCHEMBL11542769 0.85 SLC18A3 (0.43) DRD2
Hydrochloric Acid SCHEMBL11541416 0.81 DRD1 (0.56) SIGMAR1DRD2
Hydrochloric Acid SCHEMBL11543140 0.78 DRD1 (0.51) DRD2
Iodide SCHEMBL5179692 0.70 SIGMAR1 (0.44) SIGMAR1SLC6A3GRIN1GRIN2BACHE
SCHEMBL9466471 0.69 ACHE (0.54) SIGMAR1SLC6A3ACHE
SCHEMBL486687 0.68 SLC6A3 (0.66) SIGMAR1SLC6A3ACHEDRD2
SCHEMBL8108965 0.68 SLC6A3 (0.66) SIGMAR1SLC6A3ACHEDRD2
SCHEMBL1400959 0.67 TACR1 (0.61) SIGMAR1GRIN1GRIN2BACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4172890-A CARDIOVASCULAR, PARKINSON'S DISEASE, DOPAMINERGIC SMITHKLINE CORPORATION (US) 1979-10-30 US disclosed
US-4108989-A TREATING PARKINSON*S DISEASE, CARDIOVASCULAR DISORDERS SMITHKLINE CORPORATION (US) 1978-08-22 US disclosed