SCHEMBL11545309

SCHEMBL11545309

NC(=O)c1ccc(OCCNCC(O)COc2ccccc2)nc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB1 P08588 5/20 0.58
ADRB3 P13945 5/20 0.58
ADRB2 P07550 3/20 0.58
CYP1A2 P05177 1/20 0.58
ATM Q13315 1/20 0.56
CYP3A4 P08684 1/20 0.51
CYP2D6 P10635 1/20 0.51
OPRM1 P35372 5/20 0.49
OPRD1 P41143 5/20 0.49
OPRK1 P41145 4/20 0.49
ABCB1 P08183 2/20 0.49
MEN1 O00255 1/20 0.49
KMT2A Q03164 1/20 0.49
GRIN2D O15399 1/20 0.47
GRIN3B O60391 1/20 0.47
SLC6A2 P23975 1/20 0.47
SLC6A3 Q01959 1/20 0.47
GRIN1 Q05586 1/20 0.47
KCNH2 Q12809 1/20 0.47
GRIN2A Q12879 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11546769 0.90 ADRB3 (0.51) ADRB1ADRB3ADRB2CYP1A2ATM
SCHEMBL11549703 0.86 ADRB2 (0.55) ADRB1ADRB3ADRB2CYP3A4OPRM1
SCHEMBL11545703 0.85 ADRB1 (0.45) ADRB1ADRB3ADRB2MEN1KMT2A
SCHEMBL11545627 0.85 KDM4E (0.53) ADRB1ADRB3ADRB2ATMABCB1
SCHEMBL11547605 0.83 OPRM1 (0.46) ADRB1ADRB3ADRB2CYP1A2ATM
SCHEMBL11549323 0.83 KDM4E (0.49) ADRB1ADRB3ADRB2ABCB1KMT2A
SCHEMBL11546599 0.82 ADRB2 (0.47) ADRB1ADRB3ADRB2CYP1A2CYP3A4
SCHEMBL11549418 0.81 ADRB2 (0.48) ADRB1ADRB3ADRB2CYP1A2ATM
SCHEMBL7410486 0.79 ADRB2 (0.54) ADRB1ADRB3ADRB2CYP3A4OPRM1
SCHEMBL9685167 0.78 ADRB1 (0.69) ADRB1ADRB3ADRB2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4027027-A BETA-RECEPTOR-BLOCKERS, HYPOTENSIVES AND VALODILATORS; FOR TREATING ARRYTHMIAS AND ANGINA PECTORIS CIBA-GEIGY CORPORATION (US) 1977-05-31 US claimed
US-4139623-A HYPOTENSIVE AGENTS C-G CORP. (US) 1979-02-13 US disclosed
US-4027027-A BETA-RECEPTOR-BLOCKERS, HYPOTENSIVES AND VALODILATORS; FOR TREATING ARRYTHMIAS AND ANGINA PECTORIS CIBA-GEIGY CORPORATION (US) 1977-05-31 US disclosed