SCHEMBL11545374

SCHEMBL11545374

NC(=O)c1ccc(OCCN(Cc2ccccc2)CC(O)COc2ccccc2)nc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.53
MAPT P10636 2/20 0.53
CYP1A2 P05177 1/20 0.53
CYP2D6 P10635 1/20 0.53
CYP2C9 P11712 1/20 0.53
CYP2C19 P33261 1/20 0.53
NPSR1 Q6W5P4 1/20 0.53
POLB P06746 2/20 0.51
GAA P10253 1/20 0.49
MAPK1 P28482 1/20 0.49
TSHR P16473 1/20 0.46
OPRM1 P35372 7/20 0.44
OPRD1 P41143 6/20 0.44
OPRK1 P41145 6/20 0.44
KCNH2 Q12809 2/20 0.41
GRIN2D O15399 1/20 0.41
GRIN3B O60391 1/20 0.41
SLC6A2 P23975 1/20 0.41
SLC6A3 Q01959 1/20 0.41
GRIN1 Q05586 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11546850 0.94 ALDH1A1 (0.52) ALDH1A1MAPTCYP1A2CYP2D6CYP2C9
SCHEMBL11548958 0.89 POLB (0.57) ALDH1A1MAPTCYP1A2CYP2D6CYP2C9
SCHEMBL11548610 0.88 POLB (0.47) ALDH1A1MAPTCYP1A2CYP2D6CYP2C9
SCHEMBL11546206 0.85 OPRM1 (0.52) OPRM1OPRD1OPRK1KCNH2GRIN2D
SCHEMBL11547011 0.84 POLB (0.42) ALDH1A1MAPTCYP1A2CYP2D6CYP2C9
SCHEMBL11549384 0.83 POLB (0.47) ALDH1A1MAPTCYP1A2CYP2D6CYP2C9
SCHEMBL11552589 0.81 ALDH1A1 (0.54) ALDH1A1MAPTCYP1A2CYP2D6CYP2C9
Hydrochloric Acid SCHEMBL11548608 0.80 ALDH1A1 (0.56) ALDH1A1MAPTCYP1A2CYP2D6CYP2C9
SCHEMBL9835890 0.79 ALDH1A1 (0.56) ALDH1A1MAPTCYP1A2CYP2D6CYP2C9
SCHEMBL11546317 0.77 ALDH1A1 (0.52) ALDH1A1MAPTCYP1A2CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4139623-A HYPOTENSIVE AGENTS C-G CORP. (US) 1979-02-13 US disclosed
US-4027027-A BETA-RECEPTOR-BLOCKERS, HYPOTENSIVES AND VALODILATORS; FOR TREATING ARRYTHMIAS AND ANGINA PECTORIS CIBA-GEIGY CORPORATION (US) 1977-05-31 US disclosed