SCHEMBL11548958

SCHEMBL11548958

COc1ccccc1OCC(O)CN(CCOc1ccc(C(N)=O)cn1)Cc1ccccc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.57
ALDH1A1 P00352 3/20 0.46
CYP1A2 P05177 2/20 0.46
MAPT P10636 2/20 0.46
CYP2D6 P10635 1/20 0.46
CYP2C9 P11712 1/20 0.46
CYP2C19 P33261 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
TSHR P16473 2/20 0.43
KDM4E B2RXH2 1/20 0.43
LMNA P02545 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
NNMT P40261 1/20 0.42
NR1H3 Q13133 1/20 0.42
ABCB1 P08183 4/20 0.40
GAA P10253 1/20 0.40
MAPK1 P28482 1/20 0.40
OPRM1 P35372 1/20 0.40
OPRD1 P41143 1/20 0.40
OPRK1 P41145 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11548610 0.92 POLB (0.47) POLBALDH1A1CYP1A2MAPTCYP2D6
SCHEMBL11545374 0.89 ALDH1A1 (0.53) POLBALDH1A1CYP1A2MAPTCYP2D6
SCHEMBL11549384 0.88 POLB (0.47) POLBALDH1A1CYP1A2MAPTCYP2D6
SCHEMBL11547011 0.86 POLB (0.42) POLBALDH1A1CYP1A2MAPTCYP2D6
SCHEMBL11546850 0.85 ALDH1A1 (0.52) POLBALDH1A1CYP1A2MAPTCYP2D6
SCHEMBL11546206 0.82 OPRM1 (0.52) NNMTOPRM1OPRD1OPRK1
SCHEMBL11549703 0.77 ADRB2 (0.55) MAPTKDM4ELMNAABCB1GAA
Methyl Alcohol SCHEMBL11168835 0.77 ALDH1A1 (0.53) POLBALDH1A1CYP1A2MAPTCYP2D6
SCHEMBL13916263 0.76 POLB (0.49) POLBALDH1A1CYP1A2MAPTTSHR
SCHEMBL11546634 0.75 POLB (0.44) POLBALDH1A1CYP1A2MAPTCYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4139623-A HYPOTENSIVE AGENTS C-G CORP. (US) 1979-02-13 US disclosed
US-4027027-A BETA-RECEPTOR-BLOCKERS, HYPOTENSIVES AND VALODILATORS; FOR TREATING ARRYTHMIAS AND ANGINA PECTORIS CIBA-GEIGY CORPORATION (US) 1977-05-31 US disclosed