SCHEMBL11546183

SCHEMBL11546183

CCOC(=O)C1=C(N2CCCCC2)N=C(C)C(C(=O)OCC)C1c1ccccc1C#N

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 11/20 0.44
KDM4E B2RXH2 7/20 0.44
L3MBTL1 Q9Y468 6/20 0.44
HPGD P15428 4/20 0.44
LMNA P02545 2/20 0.44
TDP1 Q9NUW8 1/20 0.44
MAPT P10636 7/20 0.42
KMT2A Q03164 6/20 0.42
MEN1 O00255 5/20 0.42
NPSR1 Q6W5P4 3/20 0.38
POLB P06746 2/20 0.38
HSD17B10 Q99714 2/20 0.37
ALOX12 P18054 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
RXFP1 Q9HBX9 1/20 0.36
TSHR P16473 2/20 0.36
GAA P10253 2/20 0.36
MAPK1 P28482 2/20 0.36
CASP1 P29466 1/20 0.36
HTT P42858 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11555682 0.99 ALDH1A1 (0.44) ALDH1A1KDM4EL3MBTL1HPGDLMNA
SCHEMBL11546967 0.88 CA1 (0.42) ALDH1A1KDM4EHPGDLMNAMAPT
SCHEMBL11551313 0.85 TSHR (0.45) ALDH1A1KDM4EL3MBTL1HPGDLMNA
SCHEMBL11547775 0.84 CACNA1C (0.46) ALDH1A1KDM4EL3MBTL1TDP1KMT2A
SCHEMBL11545904 0.84 DHFR (0.48) ALDH1A1KDM4EHPGDMAPTKMT2A
SCHEMBL11547587 0.84 PKM (0.47) ALDH1A1KDM4ELMNAMAPTKMT2A
SCHEMBL11550588 0.83 CACNA1C (0.46) ALDH1A1KDM4EL3MBTL1TDP1KMT2A
SCHEMBL11547946 0.82 NPSR1 (0.45) ALDH1A1KDM4ELMNAMAPTKMT2A
SCHEMBL11552412 0.80 ANXA2 (0.39) ALDH1A1KDM4EL3MBTL1HPGDLMNA
SCHEMBL11549829 0.79 KMT2A (0.40) ALDH1A1KDM4EL3MBTL1HPGDLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4136187-A CORONARY VESSEL DILATORS BAYER AKTIENGESELLSCHAFT (DE) 1979-01-23 US claimed
US-3959292-A HYPOTENSIVE AGENTS, CORONARY DILATORS BAYER AKTIENGESELLSCHAFT (DT) 1976-05-25 US claimed
US-4136187-A CORONARY VESSEL DILATORS BAYER AKTIENGESELLSCHAFT (DE) 1979-01-23 US disclosed
US-3959292-A HYPOTENSIVE AGENTS, CORONARY DILATORS BAYER AKTIENGESELLSCHAFT (DT) 1976-05-25 US disclosed