SCHEMBL11549829

SCHEMBL11549829

CCOC(=O)C1=C(N2CCCCC2)N=C(C)C(C(=O)OCC)C1c1ccc(C)cc1S

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 5/20 0.40
MEN1 O00255 4/20 0.40
POLB P06746 1/20 0.40
HSD17B10 Q99714 3/20 0.38
ALDH1A1 P00352 8/20 0.38
KDM4E B2RXH2 4/20 0.38
MAPT P10636 4/20 0.38
SMN1; SMN2 Q16637 3/20 0.38
HPGD P15428 2/20 0.38
LMNA P02545 2/20 0.38
ALOX12 P18054 2/20 0.38
NPC1 O15118 3/20 0.36
RAB9A P51151 3/20 0.36
RXFP1 Q9HBX9 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.34
TSHR P16473 2/20 0.34
NPSR1 Q6W5P4 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11546967 0.83 CA1 (0.42) KMT2AMEN1POLBHSD17B10ALDH1A1
SCHEMBL11547775 0.82 CACNA1C (0.46) KMT2AALDH1A1KDM4EL3MBTL1NPSR1
SCHEMBL11547587 0.82 PKM (0.47) KMT2AMEN1HSD17B10ALDH1A1KDM4E
SCHEMBL11550588 0.81 CACNA1C (0.46) KMT2AALDH1A1KDM4EL3MBTL1NPSR1
SCHEMBL11551313 0.80 TSHR (0.45) KMT2AMEN1POLBHSD17B10ALDH1A1
SCHEMBL11547946 0.80 NPSR1 (0.45) KMT2AMEN1HSD17B10ALDH1A1KDM4E
SCHEMBL11545904 0.80 DHFR (0.48) KMT2AMEN1POLBHSD17B10ALDH1A1
SCHEMBL11546183 0.79 ALDH1A1 (0.44) KMT2AMEN1POLBHSD17B10ALDH1A1
SCHEMBL11555682 0.78 ALDH1A1 (0.44) KMT2AMEN1POLBHSD17B10ALDH1A1
SCHEMBL11549832 0.78 HSD17B10 (0.39) KMT2AMEN1POLBHSD17B10ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4136187-A CORONARY VESSEL DILATORS BAYER AKTIENGESELLSCHAFT (DE) 1979-01-23 US claimed
US-3959292-A HYPOTENSIVE AGENTS, CORONARY DILATORS BAYER AKTIENGESELLSCHAFT (DT) 1976-05-25 US claimed
US-4136187-A CORONARY VESSEL DILATORS BAYER AKTIENGESELLSCHAFT (DE) 1979-01-23 US disclosed
US-3959292-A HYPOTENSIVE AGENTS, CORONARY DILATORS BAYER AKTIENGESELLSCHAFT (DT) 1976-05-25 US disclosed