SCHEMBL11546196

SCHEMBL11546196

O=C(CCSC(=O)Nc1ccccc1)OC(=O)[C@@H]1CCCN1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.42
NPSR1 Q6W5P4 1/20 0.42
ELANE P08246 1/20 0.38
HTR2C P28335 1/20 0.38
HTR2B P41595 1/20 0.38
HDAC3 O15379 2/20 0.37
HDAC4 P56524 2/20 0.37
HDAC1 Q13547 2/20 0.37
HDAC7 Q8WUI4 2/20 0.37
HDAC2 Q92769 2/20 0.37
HDAC10 Q969S8 2/20 0.37
HDAC11 Q96DB2 2/20 0.37
HDAC8 Q9BY41 2/20 0.37
HDAC6 Q9UBN7 2/20 0.37
HDAC9 Q9UKV0 2/20 0.37
HDAC5 Q9UQL6 2/20 0.37
KLK7 P49862 2/20 0.37
CTSC P53634 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11549982 0.84 HTR2C (0.42) ALDH1A1HTR2CHTR2BCTSCEPHX2
SCHEMBL7379917 0.83 KMT2A (0.42) ELANEHTR2CHTR2BCTSCCYP1A2
SCHEMBL7373953 0.83 KMT2A (0.42) ELANEHTR2CHTR2BCTSCCYP1A2
SCHEMBL11544261 0.81 ELANE (0.38) ALDH1A1ELANEHTR2CHTR2BCTSC
SCHEMBL11545881 0.80 IDO1 (0.43) ELANEHTR2CHTR2BCTSCCYP1A2
SCHEMBL7373153 0.79 KMT2A (0.39) ELANEHTR2CHTR2BHDAC3HDAC4
SCHEMBL11547645 0.78 HTR2C (0.42) ELANEHTR2CHTR2BCTSCCYP1A2
SCHEMBL11549357 0.78 PRCP (0.39) HTR2CHTR2BCTSCDPP4
SCHEMBL10655597 0.77 ELANE (0.43) ALDH1A1ELANEHTR2CHTR2BCTSC
SCHEMBL11544707 0.77 SLC6A1 (0.41) ELANEHTR2CHTR2BCTSCCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4154840-A Antihypertensive pipecolic acid derivatives E. R. SQUIBB & SONS, INC. (US) 1979-05-15 US disclosed
US-4105776-A ANGIOTENSIN CONVERTING ENZYME INHIBITORS, HYPOTENSIVE AGENTS E. R. SQUIBB & SONS, INC. (US) 1978-08-08 US disclosed