SCHEMBL11547646

SCHEMBL11547646

CC(N)Cc1cccc(SC(F)(F)F)c1

nearest known ligand 0.58

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 4/20 0.58
HTR2C P28335 2/20 0.58
HTR2B P41595 2/20 0.58
PNMT P11086 2/20 0.50
SLC6A4 P31645 5/20 0.48
TAAR1 Q96RJ0 4/20 0.48
SLC6A2 P23975 3/20 0.48
MAOA P21397 2/20 0.48
SLC6A3 Q01959 2/20 0.48
SIGMAR1 Q99720 1/20 0.48
CYP2A6 P11509 1/20 0.48
ADORA2A P29274 1/20 0.48
ADORA1 P30542 1/20 0.48
CETP P11597 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL11546088 0.98 HTR2A (0.57) HTR2AHTR2CHTR2BPNMTSLC6A4
SCHEMBL17449716 0.88 HTR2A (0.44) HTR2AHTR2CHTR2BPNMTSLC6A4
SCHEMBL11544879 0.83 TAAR1 (0.50) HTR2AHTR2CHTR2BSLC6A4TAAR1
SCHEMBL935243 0.82 EPHX1 (0.44) HTR2AHTR2CHTR2BCETP
SCHEMBL11544149 0.81 SLC6A4 (0.46) HTR2AHTR2CHTR2BSLC6A4TAAR1
Tiflorex SCHEMBL2108377 0.80 SIGMAR1 (0.63) HTR2AHTR2CHTR2BSLC6A4SLC6A2
SCHEMBL11545130 0.79 SIGMAR1 (0.48) HTR2AHTR2CHTR2BSLC6A4SLC6A2
Tiflorex SCHEMBL11551709 0.79 SIGMAR1 (0.62) HTR2AHTR2CHTR2BSLC6A4SLC6A2
SCHEMBL12300586 0.79 CETP (0.41) HTR2AHTR2CHTR2BSIGMAR1CYP2A6
SCHEMBL5729617 0.79 PNMT (0.44) HTR2CPNMTTAAR1CETP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4129598-A ANOREXIGENIC AGENTS SYNTHELABO (FR) 1978-12-12 US claimed
US-4148923-A 1-(3'-Trifluoromethylthiophenyl)-2-ethylaminopropane pharmaceutical composition and method for treating obesity SYNTHELABO (FR) 1979-04-10 US disclosed
US-4129598-A ANOREXIGENIC AGENTS SYNTHELABO (FR) 1978-12-12 US disclosed
US-3965190-A ANOREXIGENIC SYNTHELABO (FR) 1976-06-22 US disclosed