Tiflorex

Tiflorex

SCHEMBL2108377

CCNC(C)Cc1cccc(SC(F)(F)F)c1

nearest known ligand 0.63

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 9/20 0.63
SLC6A4 P31645 4/20 0.63
HTR2A P28223 3/20 0.63
HTR2B P41595 3/20 0.63
ADRA2C P18825 2/20 0.63
ADRA1A P35348 2/20 0.63
DRD3 P35462 2/20 0.63
LMNA P02545 1/20 0.63
MAPT P10636 1/20 0.63
OPRK1 P41145 1/20 0.63
CYP3A4 P08684 3/20 0.43
CYP1A2 P05177 2/20 0.43
CYP2D6 P10635 2/20 0.43
TP53 P04637 1/20 0.43
TSHR P16473 1/20 0.43
CYP2C19 P33261 1/20 0.43
HTR2C P28335 2/20 0.38
USP2 O75604 2/20 0.38
NR1I2 O75469 1/20 0.38
ADRB1 P08588 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Tiflorex SCHEMBL11551709 0.99 SIGMAR1 (0.62) SIGMAR1SLC6A4HTR2AHTR2BADRA2C
SCHEMBL11547028 0.89 SIGMAR1 (0.55) SIGMAR1SLC6A4HTR2AHTR2BADRA2C
SCHEMBL11545130 0.87 SIGMAR1 (0.48) SIGMAR1SLC6A4HTR2AHTR2BADRA2C
SCHEMBL11545201 0.85 SIGMAR1 (0.50) SIGMAR1SLC6A4HTR2AHTR2BADRA2C
SCHEMBL11544879 0.85 TAAR1 (0.50) SIGMAR1SLC6A4HTR2AHTR2BADRA2C
SCHEMBL11544149 0.84 SLC6A4 (0.46) SIGMAR1SLC6A4HTR2AHTR2BADRA2C
SCHEMBL17449716 0.82 HTR2A (0.44) SIGMAR1SLC6A4HTR2AHTR2BADRA2C
SCHEMBL11547646 0.80 HTR2A (0.58) SIGMAR1SLC6A4HTR2AHTR2BHTR2C
Hydrochloric Acid SCHEMBL11546088 0.79 HTR2A (0.57) SIGMAR1SLC6A4HTR2AHTR2BHTR2C
Levofenfluramine SCHEMBL162006 0.78 SLC6A4 (1.00) SIGMAR1SLC6A4HTR2AHTR2BADRA2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 86 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20200060997-A1 TARR Receptor Agonists for Sexual Dysfunction JOHN MCCOY 2020-02-27 US claimed
WO-2016151295-A1 FLUORINATION PROCESS OXFORD UNIVERSITY INNOVATION LIMITED (GB) 2016-09-29 WO claimed
US-9016221-B2 Surface topographies for non-toxic bioadhesion control UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INC. (US) 2015-04-28 US claimed
US-20100226943-A1 SURFACE TOPOGRAPHIES FOR NON-TOXIC BIOADHESION CONTROL UNIVERSITY OF FLORIDA (US) 2010-09-09 US claimed
US-20100172916-A1 SUBSTITUTED HYDROXYPHENYLAMINE COMPOUNDS AUSPEX PHARMACEUTICALS, INC. (US) 2010-07-08 US claimed
WO-2010054286-A2 SUBSTITUTED HYDROXYPHENYLAMINE COMPOUNDS AUSPEX PHARMACEUTICALS, INC. (US) 2010-05-14 WO claimed
EP-1954244-A1 LYOPHILIZATION PROCESS AND PRODUCTS OBTAINED THEREBY Scidose, Llc (US) 2008-08-13 EP claimed
WO-2007061529-A1 LYOPHILIZATION PROCESS AND PRODUCTS OBTAINED THEREBY SCIDOSE LLC. (US) 2007-05-31 WO claimed
US-20070116729-A1 Lyophilization process and products obtained thereby SCIDOSE LLC 2007-05-24 US claimed
US-4148923-A 1-(3'-Trifluoromethylthiophenyl)-2-ethylaminopropane pharmaceutical composition and method for treating obesity SYNTHELABO (FR) 1979-04-10 US claimed
US-4129598-A ANOREXIGENIC AGENTS SYNTHELABO (FR) 1978-12-12 US claimed
WO-2026106796-A1 SYSTEM AND METHOD FOR THE TREATMENT OF TELOGEN EFFLUVIUM, ANDROGENETIC ALOPECIA, AND OTHER HAIR LOSS DISORDERS FOLLEA INTERNATIONAL (US) 2026-05-21 WO disclosed
WO-2026107229-A1 REDUCING THE ADDICTIVE LIABILITY OF OPIOID ANALGESICS BY CO- ADMINISTERING 5HT2 RECEPTOR AGONISTS THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY (US) 2026-05-21 WO disclosed
US-20260041652-A1 SYSTEM AND METHOD FOR PREVENTING ALOPECIA FOLLEA INT (US) 2026-02-12 US disclosed
EP-4079311-B1 NMN AND DERIVATIVES FOR USE IN THE TREATMENT OF DEPRESSION AND/OR ANXIETY IN PATIENTS HAVING A FORM OF PARKINSONISM NUVAMID SA (CH) 2025-10-01 EP disclosed
WO-1994021244-A1 METHOD OF TREATING ADDICTIVE BEHAVIORS HITZIG PIETR (US) 1994-09-29 WO disclosed
US-4148923-A 1-(3'-Trifluoromethylthiophenyl)-2-ethylaminopropane pharmaceutical composition and method for treating obesity SYNTHELABO (FR) 1979-04-10 US disclosed
US-4148923-A 1-(3'-Trifluoromethylthiophenyl)-2-ethylaminopropane pharmaceutical composition and method for treating obesity SYNTHELABO (FR) 1979-04-10 US disclosed
US-4129598-A ANOREXIGENIC AGENTS SYNTHELABO (FR) 1978-12-12 US disclosed
US-3965190-A ANOREXIGENIC SYNTHELABO (FR) 1976-06-22 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100172916-A1 SUBSTITUTED HYDROXYPHENYLAMINE COMPOUNDS MC1R, TYR, MITF SIGMAR1 773/4885SLC6A4 93/4885HTR2A 62/4885
US-20260041652-A1 SYSTEM AND METHOD FOR PREVENTING ALOPECIA DYRK4, DYRK2, STRA6 SIGMAR1 4868/4885SLC6A4 56/4885HTR2A 174/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.