SCHEMBL11550848

SCHEMBL11550848

COCCc1ccccc1OCC(O)CNCCOc1ccc(C(N)=O)cc1

nearest known ligand 0.54

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.54
CYP2D6 P10635 1/20 0.54
ATM Q13315 1/20 0.52
ADRB2 P07550 8/20 0.51
ADRB1 P08588 6/20 0.51
ADRB3 P13945 4/20 0.51
CYP1A2 P05177 1/20 0.51
KMT2A Q03164 2/20 0.50
KDM4E B2RXH2 1/20 0.50
ALDH1A1 P00352 1/20 0.50
MEN1 O00255 1/20 0.49
ABCB1 P08183 2/20 0.45
HTR1A P08908 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Tolamolol SCHEMBL611643 0.85 ATM (0.59) CYP3A4CYP2D6ATMADRB2ADRB1
Tolamolol SCHEMBL613511 0.85 ATM (0.59) CYP3A4CYP2D6ATMADRB2ADRB1
SCHEMBL11541226 0.84 ADRB2 (0.64) CYP2D6ATMADRB2ADRB1ADRB3
SCHEMBL11542670 0.84 CYP3A4 (0.72) CYP3A4CYP2D6ATMADRB2ADRB1
Tolamolol SCHEMBL8057907 0.84 ATM (0.58) CYP3A4CYP2D6ATMADRB2ADRB1
SCHEMBL11543785 0.83 ADRB2 (0.56) CYP3A4CYP2D6ATMADRB2ADRB1
SCHEMBL11545485 0.79 ADRB2 (0.51) CYP3A4CYP2D6ATMADRB2ADRB1
SCHEMBL11543422 0.78 ADRB1 (0.53) CYP3A4CYP2D6ATMADRB2ADRB1
SCHEMBL11546599 0.78 ADRB2 (0.47) CYP3A4CYP2D6ADRB2ADRB1ADRB3
SCHEMBL11544543 0.78 CYP3A4 (0.58) CYP3A4CYP2D6ATMADRB2ADRB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4165384-A ADRENERGIC BLOCKING AGENTS, CARDIOVASCULAR DISORDERS AKTIEBOLAGET HASSLE (SE) 1979-08-21 US disclosed