SCHEMBL11566176

SCHEMBL11566176

O=C(O)C1(Nc2ccc(F)cc2)CCN(Cc2ccccc2)CC1

nearest known ligand 0.60

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
FAAH O00519 1/20 0.55
OPRM1 P35372 1/20 0.54
OPRD1 P41143 1/20 0.54
OPRK1 P41145 1/20 0.54
NPFFR1 Q9GZQ6 1/20 0.54
NPFFR2 Q9Y5X5 1/20 0.54
ALDH1A1 P00352 2/20 0.51
CYP2D6 P10635 1/20 0.51
SIGMAR1 Q99720 3/20 0.50
CACNA1G O43497 3/20 0.50
GAA P10253 1/20 0.50
L3MBTL1 Q9Y468 1/20 0.50
SLC6A12 P48065 1/20 0.50
TMEM97 Q5BJF2 1/20 0.50
MCHR1 Q99705 1/20 0.50
MEN1 O00255 1/20 0.49
KMT2A Q03164 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2985624 0.91 NPFFR1 (0.62) FAAHOPRM1OPRD1OPRK1NPFFR1
SCHEMBL5556286 0.90 ALDH1A1 (0.61) FAAHOPRM1OPRD1OPRK1NPFFR1
SCHEMBL6045494 0.89 NPFFR1 (0.61) FAAHOPRM1OPRD1OPRK1NPFFR1
Hydrochloric Acid SCHEMBL11455282 0.89 NPFFR1 (0.61) FAAHOPRM1OPRD1OPRK1NPFFR1
Hydrochloric Acid SCHEMBL5240984 0.89 NPFFR1 (0.61) FAAHOPRM1OPRD1OPRK1NPFFR1
SCHEMBL11566839 0.88 OPRM1 (0.53) FAAHOPRM1OPRD1OPRK1NPFFR1
SCHEMBL11564776 0.88 CA12 (0.55) OPRM1NPFFR1NPFFR2SIGMAR1TMEM97
SCHEMBL11567112 0.87 FAAH (0.55) FAAHOPRM1OPRD1OPRK1NPFFR1
SCHEMBL11563209 0.85 OPRM1 (0.55) OPRM1OPRD1OPRK1NPFFR1NPFFR2
Hydrochloric Acid SCHEMBL11566542 0.84 OPRM1 (0.54) OPRM1OPRD1OPRK1NPFFR1NPFFR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1081635-C Substituted pyrrolidin-3-Yl-alkyl-piperidines useful as tachykinin antagonists MERRELL DOW PHARMA (US) 2002-03-27 CN disclosed
CN-1124961-A Substituted pyrrolidin-3-Yl-alkyl-piperidines useful as tachykinin antagonists MERRELL DOW PHARMA (US) 1996-06-19 CN disclosed
US-4179569-A ANALGESIC INTERMEDIATES JANSSEN PHARMACEUTICA N.V. (BE) 1979-12-18 US disclosed
US-3998834-A ANALGESICS JANSSEN PHARMACEUTICA N.V. (BE) 1976-12-21 US disclosed