SCHEMBL11574136

SCHEMBL11574136

C=CC(N)C1C=Cc2ccccc21

nearest known ligand 0.36

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 1/20 0.36
HTR6 P50406 1/20 0.36
BRD4 O60885 1/20 0.30
CCL2 P13500 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2527441 0.79 HTR6 (0.33) HTR2AHTR6
SCHEMBL11575783 0.76 HTR6 (0.31) HTR2AHTR6
SCHEMBL9056494 0.75 HTR2A (0.38) HTR2AHTR6BRD4CCL2
SCHEMBL9568818 0.72 HTR2A (0.32) HTR2A
SCHEMBL11124550 0.71 HTR2A (0.33) HTR2A
SCHEMBL29603716 0.71 SIGMAR1 (0.38) HTR2AHTR6BRD4CCL2
SCHEMBL8368203 0.71 HTR2A (0.38) HTR2AHTR6BRD4CCL2
SCHEMBL29658875 0.71 SIGMAR1 (0.41) HTR2AHTR6BRD4CCL2
SCHEMBL6752383 0.71 HTR2A (0.38) HTR2AHTR6BRD4CCL2
SCHEMBL668104 0.71 SIGMAR1 (0.38) HTR2AHTR6BRD4CCL2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4173633-A DIURETICS CIBA-GEIGY CORPORATION (US) 1979-11-06 US disclosed
US-4172945-A HYPOTENSIVE AGENTS E. R. SQUIBB & SONS, INC. (US) 1979-10-30 US disclosed
US-4138497-A Indanpentol derivatives for treating hypertension E. R. SQUIBB & SONS, INC. (US) 1979-02-06 US disclosed
US-4127578-A Diene intermediates for indantetrols E. R. SQUIBB & SONS, INC. (US) 1978-11-28 US disclosed
US-4092318-A HYPOTENSIVES E. R. SQUIBB & SONS, INC. (US) 1978-05-30 US disclosed
US-4053596-A HYPOTENSIVE AGENTS E. R. SQUIBB & SONS, INC. (US) 1977-10-11 US disclosed
US-4044040-A HYPERTENSIVE AGENTS E. R. SQUIBB & SONS, INC. (US) 1977-08-23 US disclosed