SCHEMBL11577641

SCHEMBL11577641

COC(=O)Cc1cc(C)ccc1Sc1ccc(C)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 6/20 0.50
ALDH1A1 P00352 6/20 0.50
HPGD P15428 3/20 0.50
MAPK1 P28482 3/20 0.50
KDM4E B2RXH2 2/20 0.50
ALOX15 P16050 2/20 0.50
HSD17B10 Q99714 2/20 0.50
L3MBTL1 Q9Y468 2/20 0.50
LMNA P02545 1/20 0.50
PKM P14618 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
JAK2 O60674 1/20 0.42
TP53 P04637 3/20 0.42
AGBL2 Q5U5Z8 1/20 0.41
MEN1 O00255 3/20 0.41
KMT2A Q03164 3/20 0.41
ICAM1 P05362 2/20 0.41
SELE P16581 2/20 0.41
VCAM1 P19320 2/20 0.41
MMP2 P08253 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11576701 0.83 AGBL2 (0.57) MAPTALDH1A1HPGDMAPK1KDM4E
SCHEMBL9911235 0.77 HSP90AB1 (0.44) MAPTALDH1A1HPGDKDM4EHSD17B10
SCHEMBL11759118 0.77 AGBL2 (0.53) MAPTALDH1A1HPGDALOX15PKM
SCHEMBL7708631 0.76 L3MBTL1 (0.45) MAPTALDH1A1HPGDMAPK1KDM4E
SCHEMBL11578003 0.76 MAPT (0.50) MAPTALDH1A1HPGDMAPK1KDM4E
SCHEMBL12650135 0.76 NPC1 (0.45) ALDH1A1HPGDKDM4EHSD17B10L3MBTL1
SCHEMBL11705979 0.76 CYP2C9 (0.54) MAPTHPGDALOX15L3MBTL1LMNA
SCHEMBL11757147 0.75 AGBL2 (0.55) HPGDPKMSMN1; SMN2AGBL2MMP2
SCHEMBL11613170 0.75 AGBL2 (0.66) MAPTALDH1A1HPGDKDM4EALOX15
SCHEMBL12646581 0.74 EGFR (0.56) ALDH1A1HPGDKDM4ETP53GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4118572-A CNS DEPRESSANTS, NEUROLEPTIC AGENTS, SCHIZOPHRENIA, TRANQUILIZERS HOFFMANN-LA ROCHE INC. (US) 1978-10-03 US disclosed
US-4105664-A Dibenz[b,f]oxepin derivatives HOFFMANN-LA ROCHE INC. (US) 1978-08-08 US disclosed
US-4100173-A DEPRESSANTS, SCHIZOPHRENIA, TRANQUILIZERS HOFFMANN-LA ROCHE INC. (US) 1978-07-11 US disclosed
US-4091023-A ANTISCHIZOPHRENIA AGENTS, TRANQUILIZERS HOFFMANN-LA ROCHE INC. (US) 1978-05-23 US disclosed
US-4032525-A CNS DEPRESSANTS, NEUROLEPTICS HOFFMANN-LA ROCHE INC. (US) 1977-06-28 US disclosed