SCHEMBL11580550

SCHEMBL11580550

N=C(NC(N)=O)Nc1ccc(I)cc1Br

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 8/20 0.37
CA2 P00918 8/20 0.37
CA9 Q16790 2/20 0.37
KIF11 P52732 1/20 0.36
PTPRC P08575 1/20 0.36
PTPN2 P17706 1/20 0.36
PTPN1 P18031 1/20 0.36
PTPRA P18433 1/20 0.36
PTPRB P23467 1/20 0.36
PTPRE P23469 1/20 0.36
PTPN6 P29350 1/20 0.36
NPC1 O15118 5/20 0.33
RAB9A P51151 5/20 0.33
NFKB1 P19838 3/20 0.33
NFKB2 Q00653 3/20 0.33
RELA Q04206 3/20 0.33
GAA P10253 1/20 0.33
MAPT P10636 1/20 0.33
SMN1; SMN2 Q16637 3/20 0.33
PLK1 P53350 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11580382 0.84 CA1 (0.38) CA1CA2CA9PTPRCPTPN2
SCHEMBL11578514 0.84 NPC1 (0.43) CA1CA2CA9KIF11NPC1
SCHEMBL11580439 0.82 CYP1A2 (0.43) CA1CA2CA9PTPRCPTPN2
SCHEMBL11579739 0.82 CXCR2 (0.43) CA1CA2CA9KIF11NPC1
SCHEMBL11580078 0.82 RAB9A (0.51) NPC1RAB9ANFKB1NFKB2RELA
SCHEMBL11581252 0.82 KIF11 (0.42) CA1CA2CA9KIF11NPC1
SCHEMBL11580526 0.82 MAP2K1 (0.47) KIF11MAP2K2MAP2K1
SCHEMBL11881815 0.80 CA1 (0.36) CA1CA2CA9KIF11PTPRC
SCHEMBL11051599 0.79 RAB9A (0.39) CA1CA2CA9PTPRCPTPN2
SCHEMBL11581488 0.79 MAPT (0.38) CA1CA2CA9KIF11NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4088785-A HYPOTENSIVE AGENTS WILLIAM H. RORER, INC. (US) 1978-05-09 US disclosed