SCHEMBL11590400

SCHEMBL11590400

CN(C)c1ccc2c(C(F)(F)F)cc(=O)n(C)c2n1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RXRA P19793 3/20 0.56
GAA P10253 1/20 0.42
AR P10275 10/20 0.40
HSD17B10 Q99714 2/20 0.37
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
ALOX15 P16050 1/20 0.37
TSHR P16473 1/20 0.37
MAPK1 P28482 1/20 0.37
HIF1A Q16665 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
PGR P06401 3/20 0.36
DDB1 Q16531 1/20 0.36
CRBN Q96SW2 1/20 0.36
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
MAPT P10636 1/20 0.35
THRB P10828 1/20 0.35
HPGD P15428 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11591247 0.80 NQO2 (0.44) RXRAGAAHSD17B10DDB1CRBN
SCHEMBL11589606 0.79 ALDH1A1 (0.54) RXRAGAAHSD17B10CYP1A2DDB1
SCHEMBL29377253 0.77 KDM4E (0.56) RXRAGAAHSD17B10MAPK1TDP1
SCHEMBL76177 0.77 KDM4E (0.56) RXRAGAAHSD17B10MAPK1TDP1
SCHEMBL5701185 0.73 CDK4 (0.41) GAAHSD17B10CYP1A2CYP3A4TSHR
SCHEMBL1772049 0.72 KDM4E (0.64) GAAARHSD17B10PGRKDM4E
Perchlorate SCHEMBL30042407 0.70 KDM4E (0.49) RXRAGAAHSD17B10CYP1A2CYP3A4
SCHEMBL21957305 0.69 AR (0.54) GAAARHSD17B10ALOX15TSHR
SCHEMBL17537351 0.69 CYP1A2 (0.49) GAAARHSD17B10CYP1A2CYP3A4
SCHEMBL1773043 0.65 KDM4E (0.48) GAAARHSD17B10PGRKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4103257-A BLUE TO NEAR ULTRAVIOLET THE UNITED STATES OF AMERICA AS REPRESENTED BY THE UNITED STATES DEPARTMENT OF ENERGY (US) 1978-07-25 US claimed