SCHEMBL11599735

SCHEMBL11599735

CN(C)CCOc1ccc(-c2c(C(=O)c3ccc(Cl)cc3)sc3ccccc23)cc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PAX8 Q06710 1/20 0.59
ITGA4 P13612 1/20 0.54
NAPEPLD Q6IQ20 1/20 0.54
GABRA1 P14867 1/20 0.48
GABRA5 P31644 1/20 0.48
HRH3 Q9Y5N1 1/20 0.47
CYP1A2 P05177 1/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2C19 P33261 1/20 0.46
HCRTR1 O43613 1/20 0.46
MAOB P27338 1/20 0.45
BLM P54132 1/20 0.45
PMP22 Q01453 1/20 0.45
ALDH1A1 P00352 1/20 0.44
MAPT P10636 1/20 0.44
ESRRG P62508 1/20 0.44
CNR1 P21554 2/20 0.43
CNR2 P34972 2/20 0.43
ESR1 P03372 2/20 0.43
ESR2 Q92731 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11599591 0.84 ITGA4 (0.68) PAX8ITGA4NAPEPLDHCRTR1MAOB
SCHEMBL11599882 0.79 GABRA1 (0.66) GABRA1GABRA5CYP1A2MAOBALDH1A1
SCHEMBL11550720 0.79 CNR1 (0.67) PAX8ITGA4NAPEPLDHCRTR1CNR1
SCHEMBL11672474 0.79 BCHE (0.54) PAX8HRH3MAOBCNR2ESR1
SCHEMBL11622183 0.79 HRH3 (0.50) PAX8HRH3CYP1A2CYP3A4CYP2C19
SCHEMBL11602188 0.78 HRH3 (0.45) PAX8ITGA4NAPEPLDHRH3CYP1A2
SCHEMBL11601813 0.78 CNR2 (0.53) MAOBCNR1CNR2ESR1ESR2
SCHEMBL4652009 0.78 CNR2 (0.75) PAX8ITGA4NAPEPLDHCRTR1CNR1
SCHEMBL5726049 0.78 HRH3 (0.68) HRH3CYP1A2CYP3A4CYP2C19BLM
SCHEMBL11732399 0.77 ALK (0.47) PAX8ITGA4NAPEPLDCNR2ESR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4075227-A NONSTEROIDAL ELI LILLY AND COMPANY (US) 1978-02-21 US disclosed