SCHEMBL11599591

SCHEMBL11599591

COc1cccc(C(=O)c2sc3ccccc3c2-c2ccc(OCCN(C)C)cc2)c1

nearest known ligand 0.68

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ITGA4 P13612 1/20 0.68
NAPEPLD Q6IQ20 1/20 0.68
PAX8 Q06710 1/20 0.62
HCRTR1 O43613 1/20 0.58
BCHE P06276 2/20 0.47
CNR1 P21554 1/20 0.44
CNR2 P34972 1/20 0.44
ESR1 P03372 3/20 0.44
ESR2 Q92731 1/20 0.44
PTPN1 P18031 2/20 0.43
MAOB P27338 1/20 0.43
TNKS O95271 2/20 0.43
EDNRA P25101 1/20 0.42
KDM4E B2RXH2 1/20 0.41
MEN1 O00255 1/20 0.41
MAPT P10636 1/20 0.41
HPGD P15428 1/20 0.41
KMT2A Q03164 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11599735 0.84 PAX8 (0.59) ITGA4NAPEPLDPAX8HCRTR1BCHE
SCHEMBL11601715 0.81 MAOA (0.51) ITGA4NAPEPLDPAX8BCHECNR1
SCHEMBL11621530 0.81 ITGA4 (0.52) ITGA4NAPEPLDPAX8HCRTR1BCHE
SCHEMBL11600977 0.80 ITGA4 (0.52) ITGA4NAPEPLDPAX8HCRTR1BCHE
SCHEMBL4652009 0.78 CNR2 (0.75) ITGA4NAPEPLDPAX8HCRTR1CNR1
SCHEMBL8340731 0.78 MAPT (0.49) ESR1MAOBKDM4EMEN1MAPT
SCHEMBL11600019 0.77 LMNA (0.47) PTPN1MAOBKDM4EMEN1MAPT
SCHEMBL11732399 0.77 ALK (0.47) ITGA4NAPEPLDPAX8BCHECNR2
SCHEMBL11547037 0.77 CNR1 (0.62) ITGA4NAPEPLDPAX8HCRTR1CNR1
SCHEMBL11550720 0.75 CNR1 (0.67) ITGA4NAPEPLDPAX8HCRTR1CNR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4075227-A NONSTEROIDAL ELI LILLY AND COMPANY (US) 1978-02-21 US disclosed