Zoledronic Acid Anhydrous

Zoledronic Acid Anhydrous

SCHEMBL1160460

O=P(O)(O)C(O)(Cn1ccnc1)P(=O)(O)O.[NaH]

nearest known ligand 0.96

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

FDPS

The experimentally established mechanism targets of Zoledronic Acid Anhydrous. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
FDPS known ✓ P14324 10/20 0.96
GGPS1 O95749 3/20 0.93
BTN3A1 O00481 1/20 0.93
CA12 O43570 1/20 0.93
CA2 P00918 1/20 0.93
LMNA P02545 1/20 0.93
MMP2 P08253 1/20 0.93
MMP9 P14780 1/20 0.93
MMP8 P22894 1/20 0.93
MMP14 P50281 1/20 0.93
CA9 Q16790 1/20 0.93
CA14 Q9ULX7 1/20 0.93
ALDH1A1 P00352 1/20 0.43
CYP11B1 P15538 1/20 0.41
CYP11B2 P19099 1/20 0.41
EGLN3 Q9H6Z9 1/20 0.41
TBXAS1 P24557 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Zoledronic Acid Anhydrous SCHEMBL3141677 1.00 FDPS (0.96) FDPSGGPS1BTN3A1CA12CA2
Zoledronic Acid Anhydrous SCHEMBL515095 1.00 FDPS (0.96) FDPSGGPS1BTN3A1CA12CA2
Zoledronic Acid Anhydrous SCHEMBL536817 0.98 FDPS (0.97) FDPSGGPS1BTN3A1CA12CA2
Zoledronic Acid Anhydrous SCHEMBL3007590 0.98 FDPS (0.97) FDPSGGPS1BTN3A1CA12CA2
Zoledronic Acid Anhydrous SCHEMBL3154439 0.98 FDPS (0.97) FDPSGGPS1BTN3A1CA12CA2
Zoledronic Acid Anhydrous SCHEMBL1586366 0.98 FDPS (1.00) FDPSGGPS1BTN3A1CA12CA2
Zoledronic Acid Anhydrous SCHEMBL19054 0.98 FDPS (1.00) FDPSGGPS1BTN3A1CA12CA2
Zoledronic Acid Anhydrous SCHEMBL22534391 0.96 FDPS (0.96) FDPSGGPS1BTN3A1CA12CA2
Zoledronic Acid Anhydrous SCHEMBL1160625 0.96 FDPS (1.00) FDPSGGPS1BTN3A1CA12CA2
Zoledronic Acid Anhydrous SCHEMBL435847 0.96 FDPS (1.00) FDPSGGPS1BTN3A1CA12CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 264 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117860968-A Bionic periosteum with bone immunoregulation function and preparation method and application thereof 中国人民解放军陆军特色医学中心 2024-04-12 CN claimed
CN-117185281-A Carbon point capable of quantitatively evaluating bone targeting performance, method for synthesizing carbon point based on chain transfer one-step method, evaluation method and application 哈尔滨工业大学 2023-12-08 CN claimed
WO-2023179588-A1 TRUNCATED VARICELLA-ZOSTER VIRUS ENVELOPE GLYCOPROTEIN GE 厦门大学 2023-09-28 WO claimed
CN-115920129-A Composite microsphere carrying water-soluble medicine and having poly dopamine layer on surface, and preparation method and application thereof 广东省科学院生物与医学工程研究所 2023-04-07 CN claimed
CN-115887783-A Polyester-based composite microsphere with calcium-phosphorus-containing layer on surface as well as preparation method and application of polyester-based composite microsphere 广东省科学院生物与医学工程研究所 2023-04-04 CN claimed
CN-115804866-A Polyester-based microsphere containing drug-loaded calcium inorganic matter and preparation method and application thereof 广东省科学院生物与医学工程研究所 2023-03-17 CN claimed
CN-114752560-B Umbilical cord mesenchymal stem cell culture medium 苏州科贝生物技术有限公司 2022-09-13 CN claimed
CN-114752560-A Umbilical cord mesenchymal stem cell culture medium 苏州科贝生物技术有限公司 2022-07-15 CN claimed
CN-110063939-B Hollow hydroxyapatite drug-loaded particle for shock wave mediated release and preparation method thereof 邢更彦 2021-08-17 CN claimed
EP-3246032-B1 PHARMACEUTICAL COMPOSITIONS COMPRISING ZOLEDRONIC ACID, CALCIUM AND VITAMIN D, SUITABLE FOR THE TREATMENT AND/OR PROPHYLAXIS OF DISEASES RELATED TO BONE METABOLISM AND OF TREATMENT-RELATED SIDE EFFECTS SUCH AS HYPOCALCAEMIA KARL CHRISTOPH (CH) 2021-08-11 EP claimed
EP-2459176-A2 CRYSTALLIZATION METHOD AND BIOAVAILABILITY Thar Pharmaceuticals, Inc. (US) 2012-06-06 EP claimed
WO-2011097269-A1 CRYSTALLIZATION METHOD AND BIOAVAILABILITY THAR PHARMACEUTICALS, INC. (US) 2011-08-11 WO claimed
CN-102070668-A Method for preparing zoledronic acid and sodium salt thereof by utilizing phase transfer catalyst BENGBU BBCA MEDICINE SCIENCE DEV CO LTD 2011-05-25 CN claimed
WO-2011014766-A2 CRYSTALLIZATION METHOD AND BIOAVAILABILITY THAR PHARMACEUTICALS, INC. (US) 2011-02-03 WO claimed
US-20110028435-A1 CRYSTALLIZATION METHOD AND BIOAVAILABILITY THAR PHARMACEUTICALS, INC. (US) 2011-02-03 US claimed
EP-1923394-A1 Reagent and use thereof for the production of bisphosphonates Sandoz A/S (DK) 2008-05-21 EP claimed
EP-1612212-A1 Zoledronic acid crystal forms, zoledronate sodium salt crystal forms, amorphous zoledronate sodium salt, and processes for their preparation Teva Pharmaceutical Industries Ltd (IL) 2006-01-04 EP claimed
EP-1567533-A2 ZOLEDRONIC ACID CRYSTAL FORMS, ZOLEDRONATE SODIUM SALT CRYSTAL FORMS, AMORPHOUS ZOLEDRONATE SODIUM SALT, AND PROCESSES FOR THEIR PREPARATION TEVA PHARMACEUTICAL INDUSTRIES LTD. (IL) 2005-08-31 EP claimed
US-20050054616-A1 Zoledronic acid crystal forms, zoledronate sodium salt crystal forms, amorphous zoledronate sodium salt, and processes for their preparation TEVA PHARMACEUTICALS USA, INC. 2005-03-10 US claimed
WO-2005005447-A2 ZOLEDRONIC ACID CRYSTAL FORMS, ZOLEDRONATE SODIUM SALT CRYSTAL FORMS, AMORPHOUS ZOLEDRONATE SODIUM SALT, AND PROCESSES FOR THEIR PREPARATION TEVA PHARMACEUTICAL INDUSTRIES LTD. (IL) 2005-01-20 WO claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050054616-A1 Zoledronic acid crystal forms, zoledronate sodium salt crystal forms, amorphous zoledronate sodium salt, and processes for their preparation SOST, FGF23, PTH1R FDPS 905/4885GGPS1 588/4885BTN3A1 1364/4885
US-20110028435-A1 CRYSTALLIZATION METHOD AND BIOAVAILABILITY PYGL, PDE8A, SLC34A1 FDPS 781/4885GGPS1 1135/4885BTN3A1 4666/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.