SCHEMBL11612464

SCHEMBL11612464

CCCCOC(=O)c1ccc2[nH]ccc2c1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 6/20 0.54
LMNA P02545 2/20 0.54
CYP1A2 P05177 2/20 0.54
TSHR P16473 2/20 0.54
CYP2C19 P33261 2/20 0.54
CYP2D6 P10635 1/20 0.54
MAPK1 P28482 1/20 0.54
NR1H2 P55055 1/20 0.54
RNASEL Q05823 1/20 0.54
SMN1; SMN2 Q16637 1/20 0.54
CYP3A4 P08684 1/20 0.52
CYP2C9 P11712 1/20 0.52
PDE4D Q08499 1/20 0.52
MAOA P21397 2/20 0.52
HPGD P15428 1/20 0.48
RECQL P46063 1/20 0.48
CTNNB1 P35222 1/20 0.48
WNT3A P56704 1/20 0.48
ACHE P22303 1/20 0.47
HTR4 Q13639 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27553735 0.95 NPC1 (0.55) ESR1MAOASTS
SCHEMBL28756834 0.90 ESR1 (0.55) ESR1LMNACYP1A2TSHRCYP2C19
SCHEMBL31094660 0.85 MAOA (0.67) ESR1CYP1A2CYP2C19MAPK1SMN1; SMN2
SCHEMBL1222893 0.85 MAOA (0.67) ESR1CYP1A2CYP2C19MAPK1SMN1; SMN2
Hydrochloric Acid SCHEMBL28263903 0.84 MAOA (0.65) CYP1A2CYP2C19MAPK1SMN1; SMN2CYP3A4
SCHEMBL709064 0.82 ESR1 (0.67) ESR1LMNACYP1A2TSHRCYP2C19
SCHEMBL14398520 0.82 TAS1R3 (0.49) CYP1A2CYP2C19CYP2D6CYP3A4MAOA
SCHEMBL4768975 0.81 HDAC1 (0.47) CYP1A2CYP2C19CYP3A4MAOACTNNB1
SCHEMBL29012860 0.81 ALDH1A1 (0.57) ESR1LMNATSHRMAOAHPGD
SCHEMBL16859558 0.81 ESR1 (0.65) ESR1LMNACYP1A2TSHRCYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100513392-C Heteroaryl substituted acetone derivatives as phospholipase A2Inhibitor of (2) MERCKLE GMBH (DE) 2009-07-15 CN disclosed
CN-1761649-A Novel heteroaryl substituted acetone derivatives as phospholipase A2Inhibitor of (2) MERCKLE GMBH (DE) 2006-04-19 CN disclosed
US-4101583-A Alpha-methylthio-alpha-(2-aminophenyl) acetaldehyde diloweralkyl acetals THE OHIO STATE UNIVERSITY RESEARCH FOUNDATION (US) 1978-07-18 US disclosed
US-4080341-A Carbazolenine and indole compounds THE OHIO STATE UNIVERSITY RESEARCH FOUNDATION (US) 1978-03-21 US disclosed
US-4067875-A Certain N-phenyl or N-pyridyl aza sulfonium salts THE OHIO STATE UNIVERSITY RESEARCH FOUNDATION (US) 1978-01-10 US disclosed
US-3992392-A Synthesis of indoles from anilines and intermediates therein THE OHIO STATE UNIVERSITY RESEARCH FOUNDATION (US) 1976-11-16 US disclosed