SCHEMBL11624409

SCHEMBL11624409

Cc1ccncc1C1=CC(=O)CCC1

nearest known ligand 0.46

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 2/20 0.40
PTGS1 P23219 1/20 0.40
CYP11B2 P19099 6/20 0.37
CYP11B1 P15538 3/20 0.37
PDE3B Q13370 1/20 0.36
PDE3A Q14432 1/20 0.36
SIGMAR1 Q99720 1/20 0.35
CYP17A1 P05093 1/20 0.35
SIRT3 Q9NTG7 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
CYP1A2 P05177 2/20 0.34
CYP2E1 P05181 2/20 0.34
CYP3A4 P08684 2/20 0.34
CYP2C8 P10632 2/20 0.34
CYP2D6 P10635 2/20 0.34
CYP2A6 P11509 2/20 0.34
CYP2C9 P11712 2/20 0.34
CYP2B6 P20813 2/20 0.34
CYP2C19 P33261 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11621375 0.87 PDE3B (0.36) PTGS2PTGS1PDE3BPDE3ASIGMAR1
SCHEMBL19371191 0.77 SIGMAR1 (0.35) SIGMAR1TDP1
SCHEMBL11620925 0.77 MEN1 (0.31)
SCHEMBL11619745 0.77 CYP11B2 (0.34) PTGS2PTGS1CYP11B2CYP11B1CYP17A1
SCHEMBL11619747 0.77 CYP11B2 (0.34) PTGS2PTGS1CYP11B2CYP11B1CYP17A1
SCHEMBL31678641 0.76 ALDH1A1 (0.39) CYP2A6
SCHEMBL11279823 0.73 MAPK14 (0.41) CYP11B2CYP11B1SIGMAR1
SCHEMBL1711669 0.73 MEN1 (0.41) CYP11B2CYP11B1
SCHEMBL11622684 0.71 NOS3 (0.32)
SCHEMBL11623144 0.71 MKNK1 (0.39) PDE3BPDE3ATDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4127583-A Preparation of 3-(pyridinyl)-2-cyclohexene-1-ones STERLING DRUG INC. (US) 1978-11-28 US disclosed
US-4111946-A Preparation of 3-(pyridinyl)-2-cyclohexen-1-ones STERLING DRUG INC. (US) 1978-09-05 US disclosed
US-4075217-A Conversion of 3-(pyridinyl)-2-cyclohexen-1-one to 3-(pyridinyl)anilines STERLING DRUG INC. (US) 1978-02-21 US disclosed
US-4026900-A 3-(Pyridinyl)-2-cyclohexen-1-ones STERLING DRUG INC. (US) 1977-05-31 US disclosed