SCHEMBL1162955

SCHEMBL1162955

CC(C)(C)c1cc(-n2cncn2)ccc1OC(N)=O

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ICAM1 P05362 1/20 0.40
SELE P16581 1/20 0.40
VCAM1 P19320 1/20 0.40
SMN1; SMN2 Q16637 2/20 0.39
MAPT P10636 2/20 0.39
HSP90AA1 P07900 1/20 0.39
HTT P42858 1/20 0.39
KDM4E B2RXH2 1/20 0.38
ALDH1A1 P00352 1/20 0.38
GPR119 Q8TDV5 2/20 0.38
MAPK10 P53779 1/20 0.38
CYP1A2 P05177 2/20 0.36
CYP2C9 P11712 2/20 0.36
CYP2C19 P33261 2/20 0.36
CYP2D6 P10635 1/20 0.36
CTSD P07339 1/20 0.35
GRM7 Q14831 1/20 0.35
CYP3A4 P08684 1/20 0.35
DPP4 P27487 1/20 0.35
GRM2 Q14416 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9943543 0.74 SMN1; SMN2 (0.51) ICAM1SELEVCAM1SMN1; SMN2MAPT
SCHEMBL8956337 0.73 ALDH1A1 (0.48) SMN1; SMN2HTTKDM4EALDH1A1CYP2C9
SCHEMBL75568 0.70 APEX1 (0.49) SMN1; SMN2MAPTKDM4EALDH1A1CYP2C19
SCHEMBL15422590 0.70 NR1H4 (0.42) SMN1; SMN2KDM4EALDH1A1
SCHEMBL15889401 0.70 SMN1; SMN2 (0.42) SMN1; SMN2MAPTHSP90AA1HTTKDM4E
SCHEMBL29185985 0.69 KDM4E (0.55) SMN1; SMN2HTTKDM4EALDH1A1
SCHEMBL29021762 0.69 RBP4 (0.47) SMN1; SMN2KDM4EALDH1A1CYP1A2CYP2C19
SCHEMBL28400912 0.69 CYP1A2 (0.42) MAPTKDM4EALDH1A1MAPK10CYP1A2
SCHEMBL8175262 0.68 CYP1A2 (0.48) ICAM1SELEVCAM1SMN1; SMN2MAPT
SCHEMBL12012872 0.67 ALDH1A1 (0.43) SMN1; SMN2MAPTHTTKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011019538-A1 SUBSTITUTED CYCLOPROPYL COMPOUNDS, COMPOSITIONS CONTAINING SUCH COMPOUNDS AND METHODS OF TREATMENT MERCK SHARP & DOHME CORP. (US) 2011-02-17 WO disclosed