SCHEMBL11630985

SCHEMBL11630985

O=C(Cl)CNc1ccsc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIK1 P39086 1/20 0.38
MARS1 P56192 2/20 0.38
CES2 O00748 1/20 0.38
CES1 P23141 1/20 0.38
HDAC1 Q13547 1/20 0.37
LCK P06239 1/20 0.36
FYN P06241 1/20 0.36
DAO P14920 1/20 0.36
RORC P51449 1/20 0.36
HPGD P15428 1/20 0.36
IDH1 O75874 1/20 0.35
NPC1 O15118 2/20 0.35
KMT2A Q03164 1/20 0.33
RAB9A P51151 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
MAPT P10636 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
NAMPT P43490 1/20 0.33
ESRRG P62508 1/20 0.33
KDR P35968 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1821169 0.82 LCK (0.42) GRIK1MARS1CES2CES1HDAC1
SCHEMBL11627985 0.75 ABAT (0.37) GRIK1MARS1CES2CES1LCK
SCHEMBL10337824 0.73 ADRA2A (0.34) NPC1
SCHEMBL25185645 0.73 CTSS (0.38) IDH1NPC1RAB9AMAPTHTT
SCHEMBL7391543 0.72 POLB (0.47) GRIK1MARS1CES2CES1HDAC1
SCHEMBL6696349 0.71 ERCC1 (0.47) HPGDNPC1KMT2ARAB9AMAPT
SCHEMBL10557721 0.71 NPC1 (0.56) GRIK1MARS1HPGDNPC1KMT2A
SCHEMBL29473470 0.70 HPGD (0.47) GRIK1MARS1CES2CES1HDAC1
SCHEMBL6715569 0.70 ALDH1A1 (0.53) HDAC1HPGDNPC1KMT2ARAB9A
SCHEMBL7432515 0.69

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4086423-A CEPHALOSPORINS, CYCLOADDITION OF GLYCINE DERIVATIVE TO THIAZINE COMPOUND MERCK & CO., INC. (US) 1978-04-25 US disclosed