SCHEMBL11632501

SCHEMBL11632501

CCc1ccc2c(c1)Cc1ccc(C#N)cc1[S+]2[O-]

nearest known ligand 0.42

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 1/20 0.42
DRD2 P14416 4/20 0.32
DRD3 P35462 4/20 0.32
SIGMAR1 Q99720 1/20 0.32
OPRD1 P41143 1/20 0.32
TRPA1 O75762 1/20 0.32
LOXL2 Q9Y4K0 1/20 0.31
PNMT P11086 1/20 0.31
NAMPT P43490 1/20 0.30
KDM4E B2RXH2 1/20 0.30
ALDH1A1 P00352 1/20 0.30
TSHR P16473 1/20 0.30
CASP1 P29466 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7044069 0.83 TRPA1 (0.36) CYP2A6TRPA1KDM4EALDH1A1
SCHEMBL166962 0.79 CYP1A2 (0.38) CYP2A6DRD2TRPA1KDM4EALDH1A1
SCHEMBL11631831 0.79 TRPA1 (0.46) DRD2DRD3TRPA1PNMTNAMPT
SCHEMBL6860681 0.76 CYP1A2 (0.38) CYP2A6DRD2TRPA1KDM4EALDH1A1
SCHEMBL11632026 0.75 ALDH1A1 (0.44) DRD3OPRD1ALDH1A1TSHRCASP1
SCHEMBL11633508 0.70
SCHEMBL5684781 0.70 CYP2A6 (0.51) CYP2A6LOXL2TSHR
SCHEMBL2308285 0.69 GAA (0.37) KDM4EALDH1A1TSHR
SCHEMBL4379538 0.68 HTR2A (0.39) DRD2DRD3ALDH1A1TSHR
SCHEMBL215978 0.68 SLC6A2 (0.31) CYP2A6ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4103015-A TRICYCLIC THIOXANTHONE-10,10-DIOXIDES BURROUGHS WELLCOME CO. (US) 1978-07-25 US disclosed